Herbicidal heterocyclic sulfonamides

ABSTRACT

This invention relates to certain heterocyclic sulfonylurea herbicidal compounds, agriculturally suitable compositions thereof and a method of their use.

BACKGROUND OF THE INVENTION

This invention relates to novel ketone pyrazole, thiophene, and pyridine sulfonylurea herbicidal compounds, agriculturally suitable compositions thereof and a method of using them to control the growth of undesired vegetation.

New compounds effective for controlling the growth of undesired vegetation are in constant demand. In the most common situation, such compounds are sought to selectively control the growth of weeds in useful crops such as cotton, rice, corn, wheat and soybeans, to name a few. Unchecked weed growth in such crops can cause significant losses, reducing profit to the farmer and increasing costs to the consumer. In other situations, herbicides are desired which will control all plant growth. Examples of areas in which complete control of all vegetation is desired are areas around fuel shortage tanks, ammunition depots and industrial storage areas. There are many products commercially available for these purposes, but the search continues for products which are more effective, less costly and environmentally safe.

The "sulfonylurea" herbicides are an extremely potent class of herbicides discovered within the last few years. A multitude of structural variations exist within the class of herbicides, but they generally consist of a sulfonylurea bridge, --SO₂ NHCONH--, linking two aromatic or heteroaromatic rings.

EP-A95,925 which was published 12/7/83 discloses herbicidal sulfonylureas of formula ##STR1## wherein

Q is, in part, ##STR2##

R₁₀ is H, C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, CO₂ R₂₄, SO₂ NR₂₀ R₂₁ or SO₂ R₂₂ ;

R₁₁ is H, C₁ -C₃ alkyl, F, Cl, Br, NO₂, OR₁₆, CO₂ R₂₄, S(O)_(m) R₂₅ or SO₂ NR₂₀ R₂₁ ; provided that when R₁₀ is other than C₁ -C₃ alkyl, then R₁₁ is H, Cl, OCH₃, NO₂, or CH₃ ;

R₁₂ is H or CH₃ ;

R₁₃ and R₁₄ are independently H, C₁ -C₃ alkyl, OR₁₆, F, Cl, Br, NO₂, CO₂ R₂₄, S(O)_(m) R₂₅ or SO₂ NR₂₀ R₂₁ ; provided that, when either of R₁₃ or R₁₄ is CO₂ R₂₄, S(O)_(m) R₂₅ or SO₂ NR₂₀ R₂₁, then the other is H, Cl, CH₃, OCH₃ or NO₂ ; and

R₁₅ is H or CH₃.

EP-A-87,780 (published 9/7/83) discloses herbicidal sulfonylureas of formula ##STR3## wherein

A is H, C₁ -C₈ alkyl or optionally substituted phenyl;

B and C are independently H, halogen, NO₂, C₁ -C₈ alkyl, arylalkyl, C₁ -C₈ alkoxy, haloalkyl, CO₂ R, CONR₁ R₂, S(O)_(n) R₃, SO₂ NR₄ R₅, or optionally substituted phenyl.

ZA 83/3850 (published 11/28/83) discloses compounds of formula ##STR4## wherein Q is a five-membered, heterocyclic radical which is bound by way of a carbon atom and contains 2 or 3 heteroatoms and which may be optionally substituted by halogen, pseudohalogen, nitro, alkyl, hydroxyl, haloalkyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, amino, alkylamino, dialkylamino, alkylcarbonylamino, alkylcarbonyl, alkoxycarbonyl, alkoxyalkyl, alkylthiocarbonyl, carbamoyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkylsulfinyl, alkylsulfonyl, alkenyloxy or alkynyloxy; and groups such as phenyl, phenoxy or phenylthio, which are unsubstituted or substituted by halogen, nitro, cyano, alkyl, alkoxy, haloalkyl, alkylcarbonyl, alkoxycarbonyl or haloalkoxy; and also benzyl unsubstituted or substituted by halogen and/or alkyl.

U.S. Pat. No. 4,127,405 and U.S. Pat. No. 4,169,719 disclose herbicidal thiophenesulfonamides, wherein the thiophene ring may be optionally substituted with CH₃, Cl or Br.

U.S. Pat. No. 4,398,939 discloses herbicidal thiophenesulfonamides, wherein the thiophene ring is substituted with substituent groups selected from C₁ -C₄ alkyl, C₃ alkenyl, OCH₃, NO₂, Cl, Br, SO₂ N(C₁ -C₃ alkyl)₂ or SO₂ N(OCH₃)CH₃.

U.S. Pat. No. 4,481,029 discloses herbicidal thiophenesulfonamides, wherein the thiophene ring is substituted with carboxylic acid, carboxylic ester and alkylcarbonyl groups or derivatives thereof.

U.S. Pat. No. 4,441,910 discloses herbicidal thiophenesulfonamides, wherein the thiophene ring is substituted with the group represented by R₆ S(O)_(n) wherein R₆ is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, cyclopentyl or cyclopropylmethyl.

European Publication No. 13,480 (published July 23, 1980) discloses herbicidal pyridine-2-, -3- and -4-sulfonylureas, wherein the pyridine ring may be substituted by Cl, Br, F, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ alkylthio, NO₂ or a carboxylic ester group.

U.S. Pat. No. 4,456,489 (issued 6/29/84) discloses herbicidal pyridine-3-sulfonylureas substituted by C₁ -C₆ alkyl-, C₃ -C₆ alkenyl-, C₂ -C₄ alkoxyalkyl- and C₅ -C₆ cycloalkylsulfonyl groups.

U.S. Pat. No. 4,518,776 (Swiss priority 7/19/82) discloses, in part, a process for the preparation of compounds of formula ##STR5## wherein

G is ##STR6##

R₁ is H, C₁ -C₄ alkyl, halogen, NO₂, CN, NH₂, S(O)_(n) C₁ -C₄ alkyl, SO₂ C₁ -C₄ alkoxy, SO₂ -di-C₁ -C₄ alkylamino, CHO, CONH₂, DC₃ -C₅ alkynyl, CODC₃ -C₅ alkynyl, DC₁ -C₄ alkyl, DC₃ -C₅ alkenyl, COC₁ -C₄ alkyl, CODC₁ -C₄ alkyl or CODC₃ -C₅ alkenyl;

n is 1 or 2;

D is O, S, NH or NC₁ -C₄ alkyl;

R₂ is H, halogen, CF₃, NO₂, C₁ -C₄ alkyl or C₁ -C₄ alkoxy; and

A is O, S, NR₅ or --C═N--.

U.S. Pat. No. 4,521,597 discloses, in part, a process for the preparation of compounds of formula ##STR7## wherein

A is ##STR8##

R₃ is H, halogen, NO₂, OCH₃ or CF₃ ;

R₅ is H, F, Cl, Br, NO₂, C₁ -C₅ alkyl, C₁ -C₅ alkoxy, CF₃, S(O)_(m) C₁ -C₅ alkyl, COR₇ or SO₂ NR₈ R₉ ;

Y is O, S, or C(R₆)═N; and

R₇ is H, C₁ -C₅ alkyl, C₁ -C₅ haloalkyl, C₁ -C₅ alkoxy, C₁ -C₅ haloalkoxy, C₂ -C₁₀ alkoxyalkoxy, C₃ -C₅ alkenyloxy, C₃ -C₅ alkynyloxy, phenoxy, benzyloxy, C₁ -C₅ alkylthio or NR₈ R₉.

U.S. Pat. No. 4,549,898 discloses herbicidal sulfonylureas of formula ##STR9## wherein

X is O, S, NR₄ or C(R₅)═N;

Y is O or S;

Z is O or S;

E is N or CH;

R₁ is H, C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkoxy, C₁ -C₄ alkoxy, halogen, C₁ -C₄ alkylthio, NR₆ R₇ or alkoxyalkyl containing not more than 4 carbon atoms;

R₂ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, NO₂, C₁ -C₃ alkoxy, C(W)R₈, SO₂ NR₆ R₇, S(O)_(n) C₁ -C₃ alkyl or COR₉ ;

R₃ is H, halogen, C₁ -C₃ alkyl, OCH₃ or CF₃ ;

R₅ is H, NO₂, F, Cl, Br, CH₃, CF₃, S(O)_(n) C₁ -C₃ alkyl, COC₁ -C₄ alkoxy or C₁ -C₃ alkoxy;

R₈ is H, C₁ -C₆ alkyl, C₁ -C₄ haloalkyl, C₃ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or alkoxyalkyl containing not more than 4 carbon atoms; and

W is O or NOR₁₀.

Japanese Patent Application No. 58-70407 (SHO 59-219,218, laid open 12/10/84) discloses pyrazole-5-sulfonylureas of formula ##STR10## wherein

A is H, lower alkyl or phenyl;

B is H or lower alkyl;

D is H, CO₂ R or COAr, halogen, NO₂ or SO₂ NR¹ R² ; and

Ar is phenyl optionally substituted with halogen.

U.S. Pat. No. 4,370,480 discloses herbicidal sulfonylureas of formula ##STR11## wherein

R₁ is ##STR12##

R is H, C₁ -C₂ alkyl, C₂ -C₆ alkenyl, C₂ -C₆ alkynyl; C₁ -C₄ alkyl substituted with one to four substituents selected from 0-3 F, 0-3 Cl, 0-3 Br, 0-2 OCH₃, 0-1 cyano, 0-1 CO₂ R₁ ' where R₁ ' is C₁ -C₃ alkyl, CO₂ R₁ ', C₂ -C₄ alkenyl substituted with 1-3 Cl, C₃ -C₆ cycloalkyl, C₅ -C₆ cycloalkenyl, C₅ -C₆ cycloalkyl substituted with substituents selected from 1-3 CH₃ or one of CH₃ CH₂, Cl, OCH₃, C₄ -C₇ cycloalkylalkyl, ##STR13## where

T₁ is ##STR14## or a single bond; and

T is O or NOR₁ ^(III).

Japanese Patent Application No. 84-273152 (Sho 86-151188, laid open July 9, 1986) discloses the following compound ##STR15##

SUMMARY OF THE INVENTION

This invention relates to novel compounds of Formula I, agriculturally suitable compositions containing them, and their method-of-use as general preemergence and/or postemergence herbicides or plant growth regulants. ##STR16## wherein

J is ##STR17##

R is H, C₁ -C₃ alkyl, phenyl, SO₂ NR_(a) R_(b), C₁ -C₂ haloalkyl, C₂ -C₄ alkoxyalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₄ alkylthioalkyl, C₂ -C₄ alkylsulfinylalkyl, C₂ -C₄ alkylsulfonylalkyl, CO₂ C₁ -C₂ alkyl, C₁ -C₄ alkylcarbonyl, C₁ -C₂ alkylsulfonyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl or C₁ -C₂ alkyl substituted with CO₂ C₁ -C₂ alkyl;

R₁ is H or CH₃ ;

R₂ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(c) R_(d), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, CO₂ R_(e), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₂ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio, CN, OH or SH;

R_(a) and R_(b) are independently C₁ -C₂ alkyl;

R_(c) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy;

R_(d) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or

R_(c) and R_(d) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --;

R_(e) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl;

R' is C₁ -C₅ alkyl, C₁ -C₅ haloalkyl, C₁ -C₅ alkyl substituted with one or two R₃ groups, C₂ -C₅ alkenyl, C₂ -C₅ haloalkenyl, C₃ -C₅ alkenyl substituted with one or two R₃ groups, C₃ -C₅ alkynyl, C₃ -C₅ haloalkynyl, C₃ -C₅ alkynyl substituted with one or two R₃ groups, C₃ -C₅ cycloalkyl, C₃ -C₅ halocycloalkyl, C₃ -C₅ cycloalkyl substituted with one or two R₄ groups, C₄ -C₇ cycloalkylalkyl, C₄ -C₇ halocycloalkylalkyl, C₄ -C₇ cycloalkylalkyl substituted with one or two R₄ groups, phenyl or benzyl;

R₃ is C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₁ -C₃ haloalkoxy, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, NO₂, OH, OR₅ or di-(C₁ -C₃ alkyl)amino;

R₄ is C₁ -C₃ alkyl, C₁ -C₃ alkoxy, C₁ -C₃ haloalkoxy, CN, NO₂, OH, OR₅ or di-(C₁ -C₃ alkyl)amino;

R₅ is SO₂ CH₃, Si(CH₃)₃, C₂ -C₃ alkylcarbonyl or CO₂ C₁ -C₂ alkyl;

E is a single bond or CH₂ ;

W is O or S;

n is 0 or 1;

n' is 0 or 1;

A is ##STR18##

X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl;

Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, ##STR19## or N(OCH₃)CH₃ ;

m is 2 or 3;

L₁ and L₂ are independently O or S;

R₆ is H or C₁ -C₃ alkyl;

R₇ and R₈ are independently C₁ -C₃ alkyl;

Z is CH or N;

Y₁ is O or CH₂ ;

X₁ is CH₃, OCH₃, OC₂ H₅ or OCF₂ H;

X₂ is CH₃, C₂ H₅ or CH₂ CF₃ ;

Y₂ is OCH₃, OC₂ H₅, SCH₃, SC₂ H₅, CH₃ or CH₂ CH₃ ;

X₃ is CH₃ or OCH₃ ;

Y₃ is H or CH₃ ;

X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl; and

Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl;

and their agriculturally suitable salts; provided that

(a) when X is Cl, F, Br or I, then Z is CH and Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃,N(CH₃)₂ or OCF₂ H;

(b) when X or Y is C₁ haloalkoxy, then Z is CH;

(c) X₄ and Y₄ are not simultaneously Cl;

(d) when W is S, then R₁ is H, A is A-1 and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or 1,3-dioxolan-2-yl;

(e) when the total number of carbons of X and Y is greater than four, then the number of carbons of R must be less than or equal to two;

(f) when J is J-1, J-2, J-3 or J-4 then R' is other than C₃ -C₅ cycloalkyl or phenyl;

(g) when J is J-5, J-6 or J-7 wherein E is a single bond, then R' is other than C₁ -C₅ alkyl, C₃ -C₅ alkenyl, phenyl, benzyl, cyclopentyl or C₄ -C₇ cycloalkylalkyl;

(h) when either or both of X and Y are OCF₂ H then J is J-1, J-2, J-3, J-4, J-8, J-9, J-10 or J-11; and

(i) when the total number of carbon atoms of X and Y is greater than four, then the total number of carbon atoms of R₂ and R' must be less than or equal to 7.

In the above definitions, the term "alkyl", used either alone or in compound words such as "alkylthio" or "haloalkyl", denotes straight chain or branched alkyl, e.g. methyl, ethyl, n-propyl, isopropyl or the different butyl and pentyl isomers.

Alkoxy denotes methoxy, ethoxy, n-propyloxy, isopropyloxy and the different butyl isomers.

Alkenyl denotes straight chain or branched alkenes, e.g., 1-propenyl, 2-propenyl, 3-propenyl and the different butenyl and pentenyl isomers.

Alkynyl denotes straight chain or branched alkynes, e.g. ethynyl, 1-propynyl, 2-propynyl and the different butynyl and pentynyl isomers.

Alkylsulfonyl denotes methylsulfonyl, ethylsulfonyl and the different propylsulfonyl isomers.

Alkylthio, alkylsulfinyl, alkylamino, etc. are defined analogously to the above examples.

Cycloalkyl denotes cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl.

The term "halogen", either alone or in compound words such as "haloalkyl", denotes fluorine, chlorine, bromine or iodine. Further, when used in compound words such as "haloalkyl" said alkyl may be partially halogenated or fully substituted with halogen atoms and said halogen atoms may be the same or different. Examples of haloalkyl include CH₂ CH₂ F, CF₂ CF₃ and CH₂ CHFCl.

The total number of carbon atoms in a substituent group is indicated by the C_(i) -C_(j) prefix where i and j are numbers from 1 to 7. For example, C₁ -C₃ alkylsulfonyl would designate methylsulfonyl through propylsulfonyl, C₂ alkoxyalkoxy would designate OCH₂ OCH₃, C₂ cyanoalkyl would designate CH₂ CN and C₃ cyanoalkyl would designate CH₂ CH₂ CN and CH(CN)CH₃.

Compounds preferred for reasons of increased ease of synthesis and/or greater herbicidal efficacy are:

1. Compounds of Formula I wherein

J is J₁ to J₁₀ and E is a single bond; or

J is J₁ to J₄ or J₈ to J₁₀ and E is CH₂ ; or

J is J₅ to J₇, E is CH₂ and

R' is C₁ -C₅ haloalkyl, C₁ -C₅ substituted with one or two R₃ groups, C₂ -C₅ alkenyl, C₂ -C₅ haloalkenyl, C₃ -C₅ alkenyl substituted with one or two R₃ groups, C₃ -C₅ alkynyl, C₃ -C₅ haloalkynyl, C₃ -C₅ alkynyl substituted with one or two R₃ groups, C₃ -C₅ cycloalkyl, C₃ -C₅ halocycloalkyl, C₃ -C₅ cycloalkyl substituted with one or two R₄ groups, C₄ -C₇ cycloalkylalkyl, C₄ -C₇ halocycloalkylalkyl, C₄ -C₇ cycloalkylalkyl substituted with one or two R₄ groups, phenyl or benzyl;

The scope of compounds within these that are first preferred can be also defined by adding the following proviso to the above described generic scope as proviso (j) when J is J-5, J-6 or J-7 and E is CH₂, then R' is other than C₁ -C₅ alkyl.

2. Compounds of Preferred 1 where E is a single bond; and W is O.

3. Compounds of Preferred 1 where E is CH₂ ; and W is O.

4. Compounds of Preferred 2 where R₂ is H, C₁ -C₃ alkyl, halogen, C₁ -C₃ alkyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br, OCH₃, SO₂ NHCH₃, SO₂ N(CH₃)₂, S(O)_(n) CH₃, CO₂ CH₃, CO₂ CH₂ CH₃, OCF₂ H, CH₂ OCH₃ or CH₂ CN;

R is H, C₁ -C₃ alkyl, phenyl, CH₂ CF₃ or CH₂ CH═CH₂ ;

X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, Cl, F, Br, I, OCF₂ H, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and

Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR20## OCF₂ H, OCF₂ Br, SCF₂ H, cyclopropyl, C.tbd.H or C.tbd.CCH₃.

5. Compounds of Preferred 4 where R' is C₁ -C₄ alkyl, C₁ -C₃ alkyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br, C₂ -C₄ alkoxyalkyl, C₂ -C₄ alkylthioalkyl, C₂ -C₄ cyanoalkyl, C₂ -C₄ alkenyl, C₂ -C₃ alkenyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br, C₃ -C₄ alkynyl, C₃ -C₅ cycloalkyl, C₃ -C₅ cycloalkyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br or cyclopropylmethyl.

6. Compounds of Preferred 5 where

A is A-1;

n is O;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃, CH(OCH₃)₂ or cyclopropyl.

7. Compounds of Preferred 6 where

R₁ is H;

R₂ is H, Cl, Br, OCH₃ or CH₃ ; and

R' is C₁ -C₃ alkyl, C₁ -C₃ alkyl substituted with 1 to 3 F, C₂ -C₃ alkoxyalkyl, C₂ -C₃ alkylthioalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₃ alkenyl, propargyl, C₃ -C₅ cycloalkyl or cyclopropylmethyl.

8. Compounds of Preferred 7 where J is J-1.

9. Compounds of Preferred 7 where J is J-2.

10. Compounds of Preferred 7 where J is J-3.

11. Compounds of Preferred 7 where J is J-4.

12. Compounds of Preferred 7 where J is J-5.

13. Compounds of Preferred 7 where J is J-6.

14. Compounds of Preferred 7 where J is J-7.

15. Compounds of Preferred 7 where J is J-8.

16. Compounds of Preferred 7 where J is J-9.

17. Compounds of Preferred 7 where J is J-10.

18. Compounds of Preferred 7 where J is J-11.

19. Compounds of Preferred 8 where R' is C₁ -C₃ alkyl.

20. Compounds of Preferred 8 where R' is C₁ -C₃ alkyl substituted with 1 to 3 F, C₂ -C₃ alkoxyalkyl, C₂ -C₃ alkylthioalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₃ alkenyl, propargyl, C₃ -C₅ cycloalkyl or cyclopropylmethyl.

21. Compounds of Preferred 3 where R is H, C₁ -C₃ alkyl, phenyl, CH₂ CF₃ or CH₂ CH═CH₂ ;

R₂ is H, Cl, Br, OCH₃ or CH₃ ;

R' is C₁ -C₃ alkyl, C₁ -C₃ alkyl substituted with 1 to 3 F, C₂ -C₃ alkoxyalkyl, C₂ -C₃ alkylthioalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₃ alkenyl, propargyl, C₃ -C₅ cycloalkyl or cyclopropylmethyl.

n is O;

A is A-1;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃, CH(OCH₃)₂ or cyclopropyl.

22. Compounds of Preferred 1 where

J is J-1, J-2, J-3 and J-4; and

R' is C₁ -C₅ haloalkyl, C₁ -C₅ alkyl substituted with one or two R₃ groups, C₂ -C₅ alkenyl, C₂ -C₅ haloalkenyl, C₃ -C₅ alkenyl substituted with one or two R₃ groups, C₃ -C₅ alkynyl, C₃ -C₅ haloalkynyl, C₃ -C₅ alkynyl substituted with one or two R₃ groups, C₃ -C₅ cycloalkyl, C₃ -C₅ halocycloalkyl, C₃ -C₅ cycloalkyl substituted with one or two R₄ groups, C₄ -C₇ cycloalkylalkyl substituted with one or two R₄ groups, phenyl or benzyl.

23. Compounds of Preferred 1 where J is J-5, J-6 or J-7.

24. Compounds of Preferred 1 where J is J-8, J-9, J-10 or J-11.

25. Compounds of Formula I wherein

J is J-5, J-6 or J-7;

E is CH₂ ; and

R' is C₁ -C₅ alkyl.

26. Compounds of Preferred 25 where when J is J-5, R₁ is H, R₂ is H, E is CH₂, A is A-1, X is OCH₃, Y is OCH₃ and Z is CH, then R' is other then CH₃.

27. Compounds of Preferred 25 where R' is C₂ -C₅ alkyl.

Specifically preferred for reasons of greatest ease of synthesis and/or greatest herbicidal efficacy are:

4-(1-oxopropyl)-N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-1H-pyrazole-5-sulfonamide, m.p. 189°-192° C.(d), and

2-(cyclopropylcarbonyl)-N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-thiophenesulfonamide, m.p. 165°-168° C.

DETAILED DESCRIPTION OF THE INVENTION Synthesis

Compounds of Formula I can be prepared by one or more of the procedures shown in Equations 1, 4, and 5. J, R₁, and A are as previously defined. ##STR21##

The reaction of Equation 1 is best carried out in an inert aprotic organic solvent such as dichloromethane, 1,2-dichloroethane, tetrahydrofuran, or acetonitrile, at a temperature between 20° and 85° C. The order of addition is not critical; however, it is often convenient to add the sulfonyl isocyanate or a solution of it in the reaction solvent, to a stirred suspension of the amine.

In some cases, the desired product is insoluble in the reaction solvent at ambient temperature and crystallizes from it in pure form. Products soluble in the reaction solvent are isolated by evaporation of the solvent. Compounds of Formula I then may be purified by trituration of the evaporation residue with solvents such as 1-chlorobutane or ethyl ether and filtration, by recrystallization from mixtures of solvents such as 1,2-dichloroethane, 1-chlorobutane and heptane or by chromatography on silica gel.

Sulfonyl isocyanates (II, W is O) are known in the art and are prepared from the corresponding sulfonamides (IV) by one of the following two general methods. ##STR22##

The sulfonamide IV is reacted with an alkyl isocyanate (e.g., n-butyl isocyanate) in a solvent whose boiling point is above 135° C., such as xylene. The reaction can optionally be carried out in the presence of a catalytic amount of 1,4-diaza[2.2.2]bicyclooctane (DABCO). The reaction mixture is heated to 135°-140° C. and held at that temperature for 5-60 minutes, after which phosgene is slowly added at such a rate that the temperature remains between 133° and 135° C. When the consumption of phosgene has ceased, the mixture is cooled and filtered to remove insoluble material. Finally, the solvent, alkyl isocyanate, and excess phosgene are evaporated, leaving the sulfonyl isocyanate (II).

If desired, the alkyl isocyanate-sulfonamide adduct can be made and isolated before reaction with the phosgene. In this case the sulfonamide (IV), alkyl isocyanate, and anhydrous base (e.g, K₂ CO₃) in a polar, aprotic solvent (e.g. acetone, butanone, or acetonitrile) are mixed and heated under reflux for 1 to 6 hours. The reaction mixture is then diluted with water, and the pH is adjusted to about 3 with acid (e.g. HCl, H₂ SO₄). The adduct is filtered out and dried, and then reacted with phosgene as described above. This procedure modification is especially useful when sulfonamide (IV) is high melting and has low solubility in the phosgenation solvent.

Sulfonyl isocyanates (II, W is O) can also be prepared by the following method. ##STR23##

The sulfonamide (IV) is heated at reflux in an excess of thionyl chloride. The reaction is continued until the sulfonamide protons are no longer detectable in the proton magnetic resonance spectrum. From 16 hours to 5 days is typically sufficient for complete conversion to the thionylamide (V) (Equation 3a).

The thionyl chloride is evaporated and the residue is treated with an inert solvent (e.g. toluene) containing at least one equivalent (typically 2-3 equivalents) of phosgene. A catalytic amount of pyridine (typically 0.1 equivalent) is added, and the mixture is heated to about 60°-140° C., with 80°-100° C. preferred. Conversion to the isocyanate (II, W is O) is usually substantially complete within 15 minutes to 3 hours (Equation 3b). The mixture is then cooled and filtered, and the solvent is evaporated, leaving the sulfonyl isocyanate (II, W is O).

Sulfonyl isothiocyanate (II, W is S) are known in the art and are prepared from the corresponding sulfonamides (IV) by reaction with carbon disulfide and potassium hydroxide followed by treatment of the resulting dipotassium salt VI with phosgene. Such a procedure is described in Arch. Pharm. 299, 174 (1966).

Many of the compounds of Formula I can be prepared by the procedure shown in Equation 4. ##STR24##

The reaction of Equation 4 is carried out by contacting phenylcarbamates or phenylthiocarbamates of Formula VI with aminoheterocycles of Formula III in an inert organic solvent such as dioxane or tetrahydrofuran at temperatures of about 20°-100° C. for a period of about one-half to twenty-four hours. The product can be isolated by evaporation of the reaction solvent and purified by methods previously described.

Phenylcarbamates and phenylthiocarbamates of Formula VI can be prepared by the methods described, or modifications thereof known to those skilled in the art, in U.S. Pat. No. 4,443,243.

Alternatively, many of the compounds of Formula I can be prepared by the method described in Equation 5. ##STR25##

The reaction of Equation 5 can be carried out by contacting equimolar amounts of a sulfonamide of Formula IV with a heterocyclic phenylcarbamate or phenylthiocarbamate of Formula VII in the presence of a base such as 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU), by methods analogous to those described in South African Patent Application 83/0441. The phenylcarbamates and phenylthiocarbamates of Formula VII can be prepared by methods, or modifications thereof known to those skilled in the art, described in South African Patent Application 82/5671 and South African Patent Application 82/5045.

The sulfonamides IV of this invention may be prepared in a variety of ways some of which are described in Equations 6 through 22.

For example, the 4-keto-5-sulfonamide isomer 1 may be prepared as outlined in Equation 6. ##STR26##

Preparation of the intermediates such as bromide 2 may be found in EPA-95,925. Exposure of bromide 2 to n-butyllithium (n-BuLi) followed by addition of the resulting anion to an acid chloride affords the protected sulfonamide. Deprotection of the sulfonamide affords the desired sulfonamide 1.

Introduction of various R and R₂ groups to sulfonamides such as 1 may be accomplished in several ways. For example, the sequence in Equation 6 could also be performed on 3-chloro-1-methylpyrazole or 1,3-dimethylpyrazole affording 3 and 4 respectively. Chloride 3 may then be used to further elaborate ##STR27## R₂ as outlined in Equation 7. ##STR28## The N-substituent of compounds such as 1, 3, 4 and 5 may also be varied by applying the same sequence of reactions as outlined in Equation 6 to various N-substituted pyrazoles. For example, pyrazole may be alkylated with dimethylsulfamoylchloride to afford pyrazole 6. Pyrazole 6 is then converted to sulfonamide 7 as outlined in Equation 8. ##STR29##

In the case where either R or R₂ are sensitive to n-BuLi (i.e. R₂ is CO₂ CH₃ or Br) then the lithiating reagent of choice is lithium diisopropylamide (LDA). Utilizing the same sequence as outlined in Equation 6 but substituting LDA for n-BuLi affords sulfonamides such as 8. This is outlined in Equation 9. ##STR30##

The isomeric 5-keto-4-sulfonamide pyrazoles may be prepared as outlined in Equations 10 and 11. ##STR31##

In Equation 10 the sequential order of group introduction is reversed to that of Equation 6. The introduction of various R and R₂ groups may be accomplished in the same manor as previously described for the 4-ketoisomer in Equations 7, 8 and 9.

An alternate synthesis of sulfonamides such as 9 is outlined in Equation 11. ##STR32##

Oxidations of alcohols to ketones such as 12 to 9 are well known in the art. For further discussion pertaining to the oxidation of alcohols to ketones, see R. H. Cornforth, J. W. Cornforth and G. Popjak, Tetrahedron, 18, 1351 (1962).

The isomeric 3-keto-4-sulfonamide such as 13 may be prepared as outlined in Equation 12. ##STR33##

In the above example of Equation 12, as before, minor variations of starting material allows for the introduction of different R and R₂ groups. The starting pyrazoles 14 or 15 may be prepared via the condensation of a hydrazine with a triketo species as outlined in Equation 13. ##STR34##

The final pyrazole isomer of the invention such as sulfonamide 16 may be prepared as outlined in Equation 14. ##STR35##

Again, as described previously, alteration of the starting material allows for the preparation of compounds such as 16 where R and/or R₂ may be varied. For example, utilizing phenylhydrazine and a chloronitrile results in pyrazole 20 and subsequently sulfonamide, 21. This is outlined in Equation 15. ##STR36##

Examples of sulfonamides which can be prepared according to Equations 6-15 are compounds 22, 23, 24, 25 and 26. ##STR37##

For further details pertaining to the synthesis of pyrazoles see EP-A-87,780, South African Patent Application 833,350, EP-A-95,925 and T. L. Jacobs, "Heterocyclic Compounds", R. C. Elderfield, ed., Vol. 5, pp. 45-161, Wiley, New York, 1957.

For further details pertaining to carbanions see J. Stowell, "Carbanions in Organic Synthesis", Wiley-Interscience, New York, 1979.

Thiophene sulfonamides such as 27 may be prepared as outlined in Equation 16. ##STR38##

Introduction of various R₂ groups on the thiophene ring may be accomplished in several ways. For example, the sequence in Equation 16 may also be performed on the 4-substituted analogs resulting in the corresponding sulfonamides such as 29 and 30. ##STR39##

The isomeric 2-thiophenesulfonamide such as 31 may be prepared as outlined in Equation 17. ##STR40##

An alternate synthesis of sulfonamides such as 31 is outlined in Equation 18. ##STR41##

The isomeric 3-thiophenesulfonamide such as 33 may be prepared as outlined in Equation 19. ##STR42##

Introduction of various R₂ groups onto the thiophene ring may be accomplished by varying the starting material as previously described.

Further details pertaining to the preparation and functional group manipulation of thiophenes may be found in U.S. Pat. No. 4,481,029.

Preparation of the pyridinesulfonamides of this invention, such as pyridine 36 may be carried out in a variety of ways. For example, Meerwein reaction of 37 followed by ortho lithiation affords sulfonamides such as 36, as outlined in Equation 20. ##STR43##

Prior to removal of the tert-butyl group it may be necessary to protect the ketone functionality as the ethylene ketal which may then be removed subsequently at a later time.

The isomeric sulfonamide, 39, may be prepared as outlined in Equation 21. ##STR44##

The isomeric sulfonamide 40 may be prepared as outlined in Equation 22. ##STR45##

Introduction of various substituents on the pyridine ring system as well as variation of R' may be accomplished as described previously for the pyrazole system.

For further details pertaining to the synthesis of pyridines see, E. Beritmaier, S. Gassenmann and E. Bayer, Tetrahedron 26, 5907 (1970); B. Blank et al., J. Med. Chem., 17, 1065 (1974); M. Mallet and G. Queguiner, Tetrahedron, 41, 3433 (1985) and J. Delarge and C. L. Lapiere, Annales Pharm. France, 36, 369 (1978).

The synthesis of heterocyclic amines such as those represented by Formula III has been reviewed in "The Chemistry of Heterocyclic Compounds," a series published by Interscience Publ., New York and London. Aminopyrimidines are described by D. J. Brown in "The Pyrimidines," Vol. XVI of the series mentioned above which is herein incorporated by reference. The 2-amino-1,3,5-triazines of Formula III, where A is A-1 and Z is N, can be prepared according to methods described by E. M. Smolin and L. Rapaport in "s-Triazines and Derivatives," vol. XIII.

Pyrimidines of Formula III, where A is A-1 and Y is an acetal or thioacetal substituent, can be prepared by methods taught in European Patent Application No. 84,224 (published July 27, 1983).

Pyrimidines of Formula III, where A is A-1 and Y is cyclopropyl or OCF₂ H can be synthesized according to the methods taught in U.S. Pat. No. 4,515,626 and U.S. Pat. No. 4,540,782, respectively.

Compounds of Formula III, where A is A-2 or A-3, can be prepared by procedures disclosed in U.S. Pat. No. 4,339,267.

Compounds of Formula III, where A is A-4, can be prepared by methods taught in U.S. Pat. No. 4,487,626.

Additional references dealing with the synthesis of bicyclic pyrimidines of Formula III, where A is A-2, A-3, or A-4 are Braker, Sheehan, Spitzmiller and Lott, J. Am. Chem. Soc., 69, 3072 (1947); Mitler and Bhattachanya, Quart. J. Indian Chem. Soc., 4, 152 (1927); Shrage and Hitchings, J. Org. Chem., 16, 1153 (1951); Caldwell, Kornfeld and Donnell, J. Am. Chem. Soc., 63, 2188 (1941); and Fissekis, Myles and Brown, J. Org. Chem., 29, 2670 (1964).

Compounds of Formula III, where A is A-5, can be prepared by methods taught in U.S. Pat. No. 4,421,550.

Compounds of Formula III, where A is A-6, can be prepared by methods taught in the U.S. Pat. No. 4,496,392.

Compounds of Formula III, where A is A-7 can be prepared by methods taught in EP-A-125,864.

Agriculturally suitable salts of compounds of Formula I are also useful herbicides and can be prepared in a number of ways known to the art. For example, metal salts can be made by contacting compounds of Formula I with a solution of an alkali or alkaline earth metal salt having a sufficiently basic anion (e.g., hydroxide, alkoxide, carbonate or hydroxide). Quaternary amine salts can be made by similar techniques.

Salts of compounds of Formula I can also be prepared by exchange of one cation for another. Cationic exchange can be effected by direct contact of an aqueous solution of a salt of a compound of Formula I (e.g., alkali or quaternary amine salt) with a solution containing the cation to be exchanged. This method is most effective when the desired salt containing the exchanged cation is insoluble in water and can be separated by filtration.

Exchange may also be effected by passing an aqueous solution of a salt of a compound of Formula I (e.g., an alkali metal or quaternary amine salt) through a column packed with a cation exchange resin containing the cation to be exchanged for that of the original salt and the desired product is eluted from the column. This method is particularly useful when the desired salt is water-soluble, e.g., a potassium sodium or calcium salt.

Acid addition salts, useful in this invention, can be obtained by reacting a compound of Formula I with a suitable acid, e.g., p-toluenesulfonic acid, trichloroacetic acid or the like.

The preparation of the compounds of this invention is further illustrated by the following specific examples. Unless otherwise indicated, temperatures are in degrees centigrade.

EXAMPLE 1 Preparation of 4-Acetyl-1-methyl-1H-pyrazole-5-sulfonamide

To a stirring solution of n-BuLi (3.7 g, 57.2 mmol) in 350 mL of tetrahydrofuran cooled to -95° C. is added 4-bromo-1-methyl-1H-pyrazole-5-t-butylsulfonamide (7.5 g, 25.4 mmol). The solution is cannulated into a stirring solution of acetyl chloride (76.2 mmol) cooled to -78° C. The reaction is stirred for 1/2 hour at -78° C. then quenched with saturated sodium chloride. The organic layer is separated, dried and concentrated. The resulting crude oil was added to CF₃ CO₂ H and allowed to stir for 24 hours. The acid was removed under vacuum and the resulting oil was flash chromatographed. The resulting solid, m.p. 153°-162° C., was mostly the closed hemiaminal, which was used directly in the next reaction.

EXAMPLE 2 Preparation of 4-Acetyl-N-[(4,6-dimethoxy-2-pyrimidinyl)aminocarbonyl]-1-methyl-1H-pyrazole-5-sulfonamide

To a mixture of the hemiaminal from Example 1 (200 mg, 0.98 mmol), the phenyl carbamate of 4,6-dimethoxy-2-aminopyrimidine (271 mg, 0.98 mmol) 3 mL of acetonitrile, and DBU (212 mg, 0.98 mmol) was added. The reaction was diluted with 3 mL of water and 3 mL of 5% hydrochloric acid. The resulting solids were collected to afford 200 mg of a white solid, m.p. 179°-182° C.; NMR (200 MHz, CDCl₃) δ 2.46 (s, 3H), 4.06 (s, 6H), 4.37 (s, 3H), 5.81 (s, 1H), 7.4 (br. s, 1H), 7.9 (s, 1H) and 13.0 (br.s, 1H); IR (KBr) 1730 cm⁻¹.

EXAMPLE 3 Preparation of N-(1,1-Dimethylethyl)-1-methyl-4-(1-oxobutyl)-1H-pyrazole-5-sulfonamide

To a solution of n-BuLi (2.1 g, 33.7 mmol) cooled to -78° C. in 250 mL of tetrahydrofuran is added the t-butyl protected 4-bromo-1-methyl-5-pyrazolesulfonamide (4.5 g, 15.2 mmol). The solution is then added to butyric anhydride (2.9 g, 18.2 mmol) at -78° C. Standard work-up afforded 4.4 g of an oil which was a mixture of the desired product and debrominated starting material. This material was not purified, but used as is in the next reaction.

EXAMPLE 4 Preparation of 1-Methyl-4-(1-oxobutyl)-1H-pyrazole-5-sulfonamide

The mixture from the previous Example 3 (3.9 g) was added to CF₃ CO₂ H (TFA) and stirred for 4.5 hours. Removal of the TFA afforded a brown oil. Flash chromatography (15:85 EtOAC:hexane (v/v)) yielded 1.0 g of a white solid, m.p. 97°-99° C. NMR (200 MHz, CDCl₃) δ 0.97 (t, 3H), 1.67 (m, 2H), 2.83 (t, 3H), 4.19 (s, 3H), 6.40 (br.s, 2H) and 7.91 (s, 1H).

EXAMPLE 5 Preparation of N-[(4-Methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]-1-methyl-4-(1-oxobutyl)-1H-pyrazole-5-sulfonamide

To a mixture of sulfonamide (150 mg, 0.61 mmol) and the phenyl carbamate of 4-methyl-6-methoxy-2-aminotriazine (158 mg, 0.61 mmol) in 3 mL of acetonitrile is added DBU (93 mg, 0.61 mmol). The solution is diluted with 3 mL of H₂ O and 3 mL of 5% HCl, and the resulting solids are collected, m.p. 174°-176° C. NMR (200 MHz, CDCl₃) δ0.88 (s, 3H), 1.68 (m, 2H), 2.7 (s, 3H), 2.79 (t, 2H), 4.19 (s, 3H), 4.33 (s, 3H), 7.7 (br.s, 1H), 7.9 (s, 1H) and 12.9 (br.s, 1H).

EXAMPLE 6 Preparation of 2-(cyclopropylcarbonyl)-N-(1-1-dimethylethyl)-3-thiophenesulfonamide

To a stirring solution of n-BuLi (6.6 g, 102 mmol) in 300 ml of tetrahydrofuran is added the t-butyl protected 3-thiophenesulfonamide (10.0 g, 45.7 mmol). The solution was warmed to -30° C. and then recooled to -78° C. The solution was cannulated into a mixture of cyclopropane carbonylic acid chloride (5.7 g, 51.7 mmol) in 50 ml of tetrahydrofuran @ -78° C. The reaction was quenched with brine, separated and dryed over magnesium sulfate, concentration of the organic in vaccuo afforded 17 g of anvil. Flash chromatography (25:75 EtCAC/hexane (v/v)) afforded 44 g of the desired product. NMR (200 MHz, CDC₃) δ1.26 (m, 13H), 2.5 (m, 1H), 6.5 (br. S, 1H), 7.5 (d, 1H), 7.67 (d, 1H):

EXAMPLE 7 Preparation of 2-(cyclopropylcarbonyl)-N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-3-thiophenesulfonamide

To a stirring solution of sulfonamide (300 mg, 1.3 mmol), the phenylcarbamate of 4,6-dimethoxy-2-aminotriazine (358 mg, 1.3 mmol) in 5 ml of acetonitrile was added DBU (197 mg, 1.3 mmol). The same work up as in example 5 afforded 390 mg of the desired product, m.p. 146°-148° C., NMR (200 mHz, CDCl₃) δ, 1.1 (m, 2H), 1.3 (m, 2H), 2.5 (m, 1H), 4.1 (S, 6H), 7.5 hr, s, 1H), 7.6 (d, 1H), 7.9 (d, 1H), 12.3 (s, 1H):

Using the procedures from Equations 1 to 22 and Examples 1 to 7 the compounds of Tables I to XIII can be prepared. ##STR46##

                                      TABLE I                                      __________________________________________________________________________     R     R.sub.1                                                                          n R.sub.2                                                                             R'         X      Y      Z  m.p. (°C.)                   __________________________________________________________________________     W = O                                                                          CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH 185-188                             CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH 180-183                             CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH 179-182                             CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N  110-112                             CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N  163-165                             CH.sub.3                                                                             H 0 H    CH.sub.3   Cl     OCH.sub.3                                                                             CH 199-201                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH 157-161                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH 151-154                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH 143-146                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub. 3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N  145-147                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N  122-137                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH 180-182                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH 163-165                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH 173-175                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH 180-184                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N  174-176                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N  154-156                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH 203-205                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub. 2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                             OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH 148-150                             CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH 178-180                             CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH 181-183                             CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N  152-154                             CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N  159-161                             CH.sub.3                                                                             H 0 H    CH(CH.sub.3).sub.2                                                                        Cl     OCH.sub.3                                                                             CH 194-196                             CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub. 2                                                              CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 F CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 F CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 F OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 F CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 F CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 F OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 F Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 F                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CHF.sub.2  CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CHF.sub.2  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CHF.sub.2  OCH.sub.3                                                                             OCH.sub. 3                                                                            CH                                     CH.sub.3                                                                             H 0 H    CHF.sub.2  CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CHF.sub.2  CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CHF.sub.2  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CHF.sub.2  Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 Cl                                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 Cl                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 Cl                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 Cl                                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 Br                                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 Br                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 Br                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 Br                                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub. 2 CH.sub.2 Br                                                                     CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 Br                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 Br                                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.2 F).sub.2                                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 I CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 I CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 I OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 I CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.3                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH(OCH.sub.3).sub.2                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(OCH.sub.3).sub.2                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(OCH.sub.3).sub.2                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SCH.sub.3                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub. 2 OCH.sub.2 F                                                                     CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OCH.sub.2 F                                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SOCH.sub.3                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 SO.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CN                                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CN                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)CN                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 NO.sub.2                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 NO.sub.2                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CN                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CN                                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OH                                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH(CH.sub.3)OH                                                                            Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 COCH.sub.3                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CO.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 N(CH.sub.3).sub.2                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH═CH.sub.2                                                                  Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH═CH.sub.2                                                                           Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 F Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CHF.sub.2  Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub. 3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 OCH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub. 3                                                                           CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH(OCH.sub.3).sub.2                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH(OCH.sub.3).sub.2                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH(OCH.sub.3).sub.2                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        CH.sub. 3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.3                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH(OCH.sub.3).sub.2                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH(OCH.sub.3).sub.2                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH(OCH.sub. 3).sub.2                                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SCH.sub.3                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub. 2 OCH.sub.2 F                                                                     Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SOCH.sub.3                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 SO.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CN                                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 CN                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH(CH.sub.3)CN                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Cl   CH.sub.2 NO.sub.2                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CH.sub.2 NO.sub.2                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CN                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Cl   CH.sub.2 CN                                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Br   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub. 2 CH.sub.3                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 OCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub. 2 CH.sub.3                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 SCH.sub.3                                                                           CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CN   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.3   OCH.sub. 3                                                                            OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub. 2 CH.sub.3                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CN   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub. 3                                                                  CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub. 2 CH.sub.3                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     H     H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      H     H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     H     H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      H     H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub. 3                                                                            N                                      H     H 0 H    CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      H     H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3).sub.2                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub. 3).sub.2                                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CH.sub.3                                                                    H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl     OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     Ph    H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      Ph    H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub. 3                                                                            N                                      Ph    H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      Ph    H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl     OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH(CH.sub.3).sub.2                                                                        Cl     OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl     OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CHF.sub.2                                                                            H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub. 2 OCH.sub.3                                                                  H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3).sub.2                                                                        Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub. 3                                                            CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 OCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 F Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.2                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CH.sub.2 F                                                                       Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  OCH.sub.3                                                                             N                                             CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CHF.sub.2  Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 CN                                                                          H 0 H    CH.sub.2 Cl                                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 Cl                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 Cl                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 CN                                                                          H 0 H    CH.sub.2 Cl                                                                               Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 Br                                                                               CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 Br                                                                               CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 Br                                                                               OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 Br                                                                               CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 Br                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 Br                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 Br                                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.3)CH.sub.2 F                                                                    Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH(CH.sub.2 F).sub.2                                                                      Cl     OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 I CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 I CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 I OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 I CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.2 SCH.sub.3                                                                   H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   H      CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   H      OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub. 3  CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                    CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH(CH.sub.3).sub.2                                                                   CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   H      OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.2 F                                                                            CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.2 F                                                                            OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCF.sub.2 H                                                                           CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCF.sub.2 H                                                                           OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.2 CF.sub.3                                                                    OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   SCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             NHCH.sub.3                                                                            N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                            N  195-197                             CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   SCF.sub.2 H                                                                           OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   Br     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.2 OCH.sub.3                                                                    OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.2 OCH.sub.3                                                                    CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   NH.sub.2                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   N(CH.sub.3).sub.2                                                                     OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   NHCH.sub.3                                                                            NHCH.sub.3                                                                            N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   cyclopropyl                                                                           OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   cyclopropyl                                                                           CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   cyclopropyl                                                                           CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   cyclopropyl                                                                           OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              CH(OCH.sub.3).sub.2                                                                   CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CF.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             C.tbd.CH                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         H      CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         H      OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                    CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH(CH.sub.3).sub.2                                                                   CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         H      OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.2 F                                                                            CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.2 F                                                                            OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCF.sub.2 H                                                                           CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCF.sub.2 H                                                                           OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.2 CF.sub.3                                                                    OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         SCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             NHCH.sub.3                                                                            N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                            N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         SCF.sub.2 H                                                                           OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         Br     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub. 2 OCH.sub.3                                                                   OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.2 OCH.sub.3                                                                    CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         NH.sub.2                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         N(CH.sub.3).sub.2                                                                     OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         NHCH.sub.3                                                                            NHCH.sub.3                                                                            N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         cyclopropyl                                                                           OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         cyclopropyl                                                                           CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         cyclopropyl                                                                           CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         cyclopropyl                                                                           OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH(OCH.sub.3).sub.2                                                                   CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CF.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             C.tbd.CH                                                                              CH                                     E is CH.sub.2                                                                  CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub. 3                                                                            OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     W = S                                                                          CH.sub. 3                                                                            H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.3   Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.3                                                                         Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub. 3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl     OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                     CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              CH.sub.3                                                                              N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                              OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                             OCH.sub.3                                                                             N                                      CH.sub.3                                                                             H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl     OCH.sub.3                                                                             CH                                     __________________________________________________________________________

                                      TABLE II                                     __________________________________________________________________________     R       R.sub.1                                                                          n R.sub.2                                                                             R'         X   Y   Z  m.p. (°C.)                       __________________________________________________________________________     CH.sub.3                                                                               H O H    CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.3   Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub. 3                                                                          N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.3                                                                         Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 F CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 F CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 F OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 F CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 F CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 F OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 F Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CHF.sub.2  CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CHF.sub.2  CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CHF.sub.2  OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CHF.sub.2  CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CHF.sub.2  CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CHF.sub.2  OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CHF.sub.2  Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 Cl                                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 Cl                                                                               CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 Cl                                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 Cl                                                                               Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.3                                                                        Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH(OCH.sub.3).sub.2                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH(OCH.sub.3).sub.2                                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH(OCH.sub.3).sub.2                                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        CH.sub. 3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 SCH.sub.3                                                                        Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 OH                                                                               Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH(CH.sub.3)OH                                                                            OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH(CH.sub.3)OH                                                                            OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub. 3                                                                              H O H    CH(CH.sub.3)OH                                                                            Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 COCH.sub.3                                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CO.sub. 2 CH.sub.3                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O H    CH.sub.2 CO.sub.2 CH.sub.3                                                                Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 N(CH.sub.3).sub.2                                                                Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH.sub.2 CH═CH.sub.2                                                                  Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.3                                                                            CH═CH.sub.2                                                                           Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH═CHOCH.sub.3                                                                        CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O Cl   CH═CHOCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH═CHOCH.sub.3                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH═CHCN                                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O Cl   CH═CHCN                                                                               CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   CH(CH.sub.3)CH═CH.sub.2                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   CH(CH.sub.3)CH═CH.sub.2                                                               Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   C.tbd.CH   CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O Cl   C.tbd.CH   CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   C.tbd.CH   OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   C.tbd.CH   CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O Cl   C.tbd.CH   CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   C.tbd.CH   OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   C.tbd.CH   Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   CH.sub.2 C.tbd.CH                                                                         Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 CH.sub.2 C.tbd.CH                                                                CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 CH.sub.2 C.tbd.CH                                                                CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 CH.sub.2 C.tbd.CH                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O Cl   CH.sub.2 CH.sub.2 C.tbd.CH                                                                CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O Cl   CH(CH.sub.3)C.tbd.CH                                                                      CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   CH(CH.sub.3)C.tbd.CH                                                                      OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O Cl   CH(CH.sub.3)C.tbd.CH                                                                      Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.3   Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.3                                                                         Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O CH.sub.2 F                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub. 2                                                                         CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.3   Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.3                                                                         Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.3                                                                               H O OCHF.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 F Cl OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CH.sub.2 F                                                                       Cl OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CHF.sub.2  Cl OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 Cl                                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 Cl                                                                               CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 CH═ CH.sub.2                                                              H O H    CH.sub.2 Cl                                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 CH═CH.sub.2                                                               H O H    CH.sub.2 Cl                                                                               Cl OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 OCH.sub. 3                                                                    H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3).sub.2                                                                        Cl OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 OCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 Br                                                                               CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 Br                                                                               CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 Br                                                                               OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 Br                                                                               CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 Br                                                                      CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 Br                                                                      OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 Br                                                                      Cl OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.3)CH.sub.2 F                                                                    Cl OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH(CH.sub.2 F).sub.2                                                                      Cl OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 I CH.sub.3                                                                          CH.sub.3                                                                            CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 I CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 I OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 I CH.sub.3                                                                          CH.sub.3                                                                            N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              CH.sub.3                                                                          OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          CH.sub.2 SCH.sub.3                                                                     H O H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              Cl OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            CH                                         Ph      H O H    CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.3   CH.sub.3                                                                          CH.sub.3                                                                            N                                          Ph      H O H    CH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.3   OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.3   Cl OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            CH                                         Ph      H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                                                                            N                                          Ph      H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.2 CH.sub.3                                                                         Cl OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          CH.sub.3                                                                            N                                          Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           CH                                         Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          CH.sub.3                                                                            N                                          Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                         OCH.sub.3                                                                           N                                          Ph      H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl OCH.sub.3                                                                           CH                                         __________________________________________________________________________

                                      TABLE III                                    __________________________________________________________________________     R    R.sub.1                                                                          n R.sub.2                                                                             R'         X   Y   Z  m.p.(°C.)                           __________________________________________________________________________     CH.sub.3                                                                            H O H    CH.sub.3   CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.3   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.3   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.3   CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.3   CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.3   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.3   Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.3                                                                         Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 Br                                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 Br                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 Br                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 Br                                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 Br                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 Br                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 Br                                                                      Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH(CH.sub.3)CH.sub.2 F                                                                    Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH(CH.sub.2 F).sub.2                                                                      Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 I CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 I CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 I OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 I CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub. 3                                                                           H O H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CH.sub.2 CH.sub.2 F                                                              Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 OH                                                                               Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            CH.sub. 3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH(CH.sub.3)OH                                                                            Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 OSi(CH.sub.3).sub.3                                                              Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 COCH.sub.3                                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O H    CH.sub.2 COCH.sub.3                                                                       CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O H    CH.sub.2 CO.sub.2 CH.sub.3                                                                Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 OCH.sub.2 F                                                                      Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                          OCH.sub.3 N                                       CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SOCH.sub.3                                                                       Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                                Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 CN                                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 CN                                                                      CH.sub. 3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 (CH.sub.3)CN                                                                     OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 NO.sub.2                                                                         CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 CH.sub.2 NO.sub.2                                                                CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 CN                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O CH.sub.3                                                                            CH.sub.2 CN                                                                               Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub. 3                                                                           H O Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH(CH.sub.3).sub.2                                                                        Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 N(CH.sub.3).sub.2                                                                Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH.sub.2 CH═CH.sub.2                                                                  Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Cl   CH═CH.sub.2                                                                           Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.3   CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Br   CH.sub.3   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub. 3                                                                           H O Br   CH.sub.3   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.3   CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Br   CH.sub.3   CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.3   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.3   Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.3                                                                         Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O Br   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub. 3  CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.3   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.3   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.3   CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.3   CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.3   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.3   Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.3                                                                         Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl  OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub. 2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           CH.sub.3                                                                           N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CH.sub.3                                                                            H O N(CH.sub.3).sub.2                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl  OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           CH.sub.3                                                                           N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl  OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           CH.sub.3                                                                           N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3).sub.2                                                                        Cl  OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl  OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           CH.sub.3                                                                           CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                            CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                             CO.sub.2 CH.sub.3                                                                   H O H    CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl  OCH.sub.3                                                                          CH                                            __________________________________________________________________________

                                      TABLE IV                                     __________________________________________________________________________     R    R.sub.1                                                                          n R.sub.2                                                                             R'        X   Y   Z  m.p. (°C.)                           __________________________________________________________________________     CH.sub.3                                                                            H 0 H    CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 H    CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 H    CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.3  Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub. 3                                                                         N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.3                                                                        Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.3                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 H    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 F                                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CH.sub.2 F                                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CHF.sub.2 Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CF.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CF.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 CF.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                              CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                              CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                              OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CH.sub.3                                                                            CH.sub.2 Cl                                                                              Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.3  Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub. 3                                                                         N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.3                                                                        Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.3                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub. 2 CH.sub.2 CH.sub.2 CH.sub.3                                                     CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 OCH.sub.3                                                                          CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   C(CH.sub.3)═CH.sub.2                                                                 Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH.sub.2 CH═CHCH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH═CH--CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CH--CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CH--CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH═CH--CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH═CH--CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH═CH--CH.sub.2 CH.sub.3                                                             Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH═CHCH.sub.2 F                                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 Cl   CH═CHF                                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.3  Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.3                                                                        Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CF.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3  CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.3  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub. 3                                                                  CH.sub.3  Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3                                                                        Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.3 CH.sub.3                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.3                                                                            H 0 CO.sub.2 CH.sub.3                                                                   CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 F                                                                               Cl  OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CH.sub.2 F                                                                      Cl  OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CHF.sub.2 Cl  OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CF.sub.3                                                                        CH.sub.3                                                                           CH.sub.3                                                                           CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CF.sub.3                                                                        CH.sub.3                                                                           OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 CF.sub.3                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                             CH.sub.2 CN                                                                         H 0 H    CH.sub.2 Cl                                                                              CH.sub.3                                                                           CH.sub.3                                                                           N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 Cl                                                                              CH.sub.3                                                                           OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 Cl                                                                              OCH.sub.3                                                                          OCH.sub.3                                                                          N                                              CH.sub.2 CN                                                                         H 0 H    CH.sub.2 Cl                                                                              Cl  OCH.sub.3                                                                          CH                                             __________________________________________________________________________

                                      TABLE V                                      __________________________________________________________________________     R.sub.1                                                                          R.sub.2                                                                             R'          X      Y      Z  m.p. (°C.)                          __________________________________________________________________________     H H    cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH 154-157                                    H H    cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH 167-171                                    H H    cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH 165-168                                    H H    cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H H    cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N  146-148                                    H H    cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N  146-149                                    H H    cyclopropyl Cl     OCH.sub.3                                                                             CH 122-125                                    H H    cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H H    cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H H    cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H H    cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H H    cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H H    cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H H    cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H H    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H H    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H H    2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H H    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H H    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H H    2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H H    2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H H    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H H    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H H    2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H H    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H H    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H H    2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H H    2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.3                                                                            cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.3                                                                            cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.3                                                                            cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.3                                                                            cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        CH.sub. 3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.3                                                                            2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H Cl   cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H Cl   cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H Cl   cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H Cl   cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H Cl   cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H Cl   cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H Cl   cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H Cl   cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H Cl   cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H Cl   cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H Cl   cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H Cl   cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H Cl   cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H Cl   cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H Cl   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H Cl   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H Cl   2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H Cl   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H Cl   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H Cl   2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H Cl   2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H Cl   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H Cl   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H Cl   2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H Cl   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H Cl   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H Cl   2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H Cl   2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H F    cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H F    cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H F    cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H F    cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H F    cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H F    cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H F    cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H F    cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H F    cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H F    cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H F    cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H F    cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H F    cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H F    cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H F    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H F    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H F    2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H F    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H F    2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H F    2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H F    2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H F    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H F    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H F    2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H F    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H F    2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H F    2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H F    2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H OCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H OCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           cyclopropyl OCH.sub. 3                                                                            OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H OCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H OCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H OCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H SCH.sub. 3                                                                          cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H SCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H SCH.sub.3                                                                           cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H SCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H SCH.sub.3                                                                           cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H SCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub. 3                                                                            CH                                            H SCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H SCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H SCH.sub.3                                                                           2.2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H SCH.sub.3                                                                           2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CO.sub.2 CH.sub.3                                                                   cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CO.sub.2 CH.sub.3                                                                   cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CO.sub.2 CH.sub.3                                                                   cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CO.sub.2 CH.sub.3                                                                   cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CO.sub.2 CH.sub.3                                                                   2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H N(CH.sub.3).sub.2                                                                   cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H N(CH.sub.3).sub.2                                                                   cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H N(CH.sub.3).sub.2                                                                   cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H N(CH.sub.3).sub.2                                                                   cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H N(CH.sub.3).sub.2                                                                   2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.2 CN                                                                         cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         cyclopropyl CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.2 CN                                                                         cyclopropyl CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         cyclopropyl OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         cyclopropyl Cl     OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.2 CN                                                                         cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         cyclobutyl  CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.2 CN                                                                         cyclobutyl  CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         cyclobutyl  OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         cyclobutyl  Cl     OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         2-fluorocyclopropyl                                                                        Cl     OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              CH                                            H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              CH.sub.3                                                                              N                                             H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                              OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                             N                                             H CH.sub.2 CN                                                                         2,2-difluorocyclopropyl                                                                    Cl     OCH.sub.3                                                                             CH                                            H H    cyclopropyl H      CH.sub.3                                                                              CH                                            H H    cyclopropyl H      OCH.sub.3                                                                             CH                                            H H    cyclopropyl CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                    CH                                            H H    cyclopropyl CH.sub.3                                                                              OCH(CH.sub.3).sub.2                                                                   CH                                            H H    cyclopropyl H      OCH.sub.3                                                                             N                                             H H    cyclopropyl OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    CH                                            H H    cyclopropyl CH.sub.2 F                                                                            CH.sub.3                                                                              CH                                            H H    cyclopropyl CH.sub.2 F                                                                            OCH.sub.3                                                                             CH                                            H H    cyclopropyl OCF.sub.2 H                                                                           CH.sub.3                                                                              CH                                            H H    cyclopropyl OCF.sub.2 H                                                                           OCH.sub.3                                                                             CH                                            H H    cyclopropyl OCH.sub.2 CF.sub.3                                                                    OCH.sub.3                                                                             N                                             H H    cyclopropyl SCH.sub.3                                                                             OCH.sub.3                                                                             CH                                            H H    cyclopropyl OCH.sub.3                                                                             NHCH.sub.3                                                                            N                                             H H    cyclopropyl OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                            N                                             H H    cyclopropyl OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    N                                             H H    cyclopropyl SCF.sub.2 H                                                                           OCH.sub.3                                                                             CH                                            H H    cyclopropyl Br     OCH.sub.3                                                                             CH                                            H H    cyclopropyl CH.sub.2 OCH.sub.3                                                                    OCH.sub.3                                                                             CH                                            H H    cyclopropyl CH.sub.2 OCH.sub.3                                                                    CH.sub.3                                                                              N                                             H H    cyclopropyl NH.sub.2                                                                              OCH.sub.3                                                                             N                                             H H    cyclopropyl N(CH.sub.3).sub.2                                                                     OCH.sub.3                                                                             N                                             H H    cyclopropyl NHCH.sub.3                                                                            NHCH.sub.3                                                                            N                                             H H    cyclopropyl cyclopropyl                                                                           OCH.sub.3                                                                             CH                                            H H    cyclopropyl cyclopropyl                                                                           CH.sub.3                                                                              N                                             H H    cyclopropyl cyclopropyl                                                                           CH.sub.3                                                                              CH                                            H H    cyclopropyl cyclopropyl                                                                           OCH.sub.3                                                                             N                                             H H    cyclopropyl CH.sub.3                                                                              CH(OCH.sub.3).sub.2                                                                   CH                                            H H    cyclopropyl CF.sub.3                                                                              OCH.sub.3                                                                             CH                                            H H    cyclopropyl OCH.sub.3                                                                             C.tbd.CH                                                                              CH                                            __________________________________________________________________________

                  TABLE VI                                                         ______________________________________                                                                                     m.p.                               R.sub.1                                                                            R.sub.2  R'            X     Y     Z    (°C.)                       ______________________________________                                         H   H        cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   H        cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   H        cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   H        cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   H        cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   H        cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   H        cyclopropyl   Cl    OCH.sub.3                                                                            CH                                      H   H        cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   H        cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   H        cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   H        cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   H        cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   H        cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   H        cyclobutyl    Cl    OCH.sub.3                                                                            CH                                      H   H        2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   H        2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   H        2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   H        2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   H        2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   H        2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   H        2-fluorocyclopropyl                                                                          Cl    OCH.sub. 3                                                                           CH                                      H   H        2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             CH                                                   propyl                                                            H   H        2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                   propyl                                                            H   H        2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                   propyl                                                            H   H        2.2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             N                                                    propyl                                                            H   H        2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            N                                                    propyl                                                            H   H        2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                    propyl                                                            H   H        2,2-difluorocyclo-                                                                           Cl    OCH.sub.3                                                                            CH                                                   propyl                                                            H   CH.sub.3 cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CH.sub.3 cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CH.sub.3 cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CH.sub.3 cycloprppyl   CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CH.sub.3 cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CH.sub.3 cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CH.sub.3 cyclopropyl   Cl    OCH.sub.3                                                                            CH                                      H   CH.sub.3 cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CH.sub.3 cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CH.sub.3 cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CH.sub.3 cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CH.sub.3 cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CH.sub.3 cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CH.sub.3 cyclobutyl    Cl    OCH.sub. 3                                                                           CH                                      H   CH.sub.3 2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CH.sub.3 2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CH.sub.3 2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CH.sub.3 2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CH.sub.3 2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CH.sub.3 2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CH.sub.3 2-fluorocyclopropyl                                                                          Cl    OCH.sub.3                                                                            CH                                      H   CH.sub.3 2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             CH                                                   propyl                                                            H   CH.sub.3 2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                   propyl                                                            H   CH.sub.3 2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                   propyl                                                            H   CH.sub.3 2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             N                                                    propyl                                                            H   CH.sub.3 2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            N                                                    propyl                                                            H   CH.sub.3 2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                    propyl                                                            H   CH.sub.3 2,2-difluorocyclo-                                                                           Cl    OCH.sub.3                                                                            CH                                                   propyl                                                            H   CH.sub.2 F                                                                              cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CH.sub.2 F                                                                              cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CH.sub.2 F                                                                              cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CH.sub.2 F                                                                              cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CH.sub.2 F                                                                              cyclopropyl   Cl    OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CH.sub.2 F                                                                              cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CH.sub.2 F                                                                              cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CH.sub.2 F                                                                              cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CH.sub.2 F                                                                              cyclobutyl    Cl    OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CH.sub.2 F                                                                              2-fluorocyclopropyl                                                                          Cl    OCH.sub.3                                                                            CH                                      H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             CH                                                   propyl                                                            H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                   propyl                                                            H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                   propyl                                                            H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             N                                                    propyl                                                            H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            N                                                    propyl                                                            H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                    propyl                                                            H   CH.sub.2 F                                                                              2,2-difluorocyclo-                                                                           Cl    OCH.sub.3                                                                            CH                                                   propyl                                                            H   OCH.sub.3                                                                               cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   OCH.sub.3                                                                               cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   OCH.sub.3                                                                               cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   OCH.sub.3                                                                               cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   OCH.sub.3                                                                               cyclopropyl   Cl    OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   OCH.sub.3                                                                               cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   OCH.sub.3                                                                               cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   OCH.sub.3                                                                               cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   OCH.sub.3                                                                               cyclobutyl    Cl    OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          CH.sub. 3                                                                            CH.sub.3                                                                             N                                       H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   OCH.sub.3                                                                               2-fluorocyclopropyl                                                                          Cl    OCH.sub.3                                                                            CH                                      H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             CH                                                   propyl                                                            H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                   propyl                                                            H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                   propyl                                                            H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             N                                                    propyl                                                            H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            N                                                    propyl                                                            H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                    propyl                                                            H   OCH.sub.3                                                                               2,2-difluorocyclo-                                                                           Cl    OCH.sub.3                                                                            CH                                                   propyl                                                            H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CO.sub.2 CH.sub.3                                                                       cyclopropyl   Cl    OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CO.sub.2 CH.sub.3                                                                       cyclobutyl    Cl    OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   CO.sub.2 CH.sub.3                                                                       2-fluorocyclopropyl                                                                          Cl    OCH.sub.3                                                                            CH                                      H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             CH                                                   propyl                                                            H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                   propyl                                                            H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                   propyl                                                            H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             N                                                    propyl                                                            H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            N                                                    propyl                                                            H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                    propyl                                                            H   CO.sub.2 CH.sub.3                                                                       2,2-difluorocyclo-                                                                           Cl    OCH.sub.3                                                                            CH                                                   propyl                                                            H   SCHF.sub.2                                                                              cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   SCHF.sub.2                                                                              cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              cyclopropyl   CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   SCHF.sub.2                                                                              cyclopropyl   CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   SCHF.sub.2                                                                              cyclopropyl   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   SCHF.sub.2                                                                              cyclopropyl   Cl    OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   SCHF.sub.2                                                                              cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              cyclobutyl    CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   SCHF.sub.2                                                                              cyclobutyl    CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   SCHF.sub.2                                                                              cyclobutyl    OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   SCHF.sub.2                                                                              cyclobutyl    Cl    OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             CH                                      H   SCHF.sub.2                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              2-fluorocyclopropyl                                                                          CH.sub.3                                                                             CH.sub.3                                                                             N                                       H   SCHF.sub. 2                                                                             2-fluorocyclopropyl                                                                          CH.sub.3                                                                             OCH.sub.3                                                                            N                                       H   SCHF.sub.2                                                                              2-fluorocyclopropyl                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                            N                                       H   SCHF.sub.2                                                                              2-fluorocyclopropyl                                                                          Cl    OCH.sub.3                                                                            CH                                      H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             CH                                                   propyl                                                            H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                   propyl                                                            H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                   propyl                                                            H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             CH.sub.3                                                                             N                                                    propyl                                                            H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           CH.sub.3                                                                             OCH.sub.3                                                                            N                                                    propyl                                                            H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                    propyl                                                            H   SCHF.sub.2                                                                              2,2-difluorocyclo-                                                                           Cl    OCH.sub.3                                                                            CH                                                   propyl                                                            ______________________________________                                    

                                      TABLE VII                                    __________________________________________________________________________                                       m.p.                                         R.sub.1                                                                           R.sub.2                                                                               R'          X   Y    Z  (°C.)                                 __________________________________________________________________________     H  H      cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  H      cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  H      cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  H      cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  H      cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  H      cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  H      cyclopropyl Cl  OCH.sub.3                                                                           CH                                              H  H      cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  H      cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  H      cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  H      cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  H      cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  H      cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  H      cyclobutyl  Cl  OCH.sub.3                                                                           CH                                              H  H      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  H      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  H      2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  H      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  H      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  H      2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  H      2-fluorocyclopropyl                                                                        Cl  OCH.sub. 3                                                                          CH                                              H  H      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  H      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  H      2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  H      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  H      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  H      2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  H      2,2-difluorocyclopropyl                                                                    Cl  OCH.sub.3                                                                           CH                                              H  Cl     cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  Cl     cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  Cl     cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  Cl     cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  Cl     cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  Cl     cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  Cl     cyclopropyl Cl  OCH.sub.3                                                                           CH                                              H  Cl     cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  Cl     cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  Cl     cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  Cl     cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  Cl     cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  Cl     cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  Cl     cyclobutyl  Cl  OCH.sub.3                                                                           CH                                              H  Cl     2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  Cl     2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  Cl     2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  Cl     2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  Cl     2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  Cl     2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  Cl     2-fluorocyclopropyl                                                                        Cl  OCH.sub.3                                                                           CH                                              H  Cl     2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  Cl     2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  Cl     2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  Cl     2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  Cl     2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  Cl     2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  Cl     2,2-difluorocyclopropyl                                                                    Cl  OCH.sub.3                                                                           CH                                              H  F      cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  F      cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  F      cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  F      cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  F      cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  F      cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  F      cyclopropyl Cl  OCH.sub.3                                                                           CH                                              H  F      cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  F      cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  F      cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  F      cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  F      cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  F      cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  F      cyclobutyl  Cl  OCH.sub.3                                                                           CH                                              H  F      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  F      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  F      2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  F      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  F      2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  F      2-fluorocyclopcopyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  F      2-fluorocyclopropyl                                                                        Cl  OCH.sub.3                                                                           CH                                              H  F      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  F      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  F      2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  F      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  F      2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  F      2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  F      2,2-difluorocyclopropyl                                                                    Cl  OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            cycloprppyl CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclopropyl Cl  OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            cyclobutyl  Cl  OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            2-fluorocyclopropyl                                                                        Cl  OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  SO.sub.2 N(CH.sub.3).sub.2                                                            2,2-difluorocyclopropyl                                                                    Cl  OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            cycloproyyl CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  OCHF.sub.2                                                                            cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  OCHF.sub.2                                                                            cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            cyclopropyl Cl  OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  OCHF.sub.2                                                                            cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  OCHF.sub.2                                                                            cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            cyclobutyl  Cl  OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  OCHF.sub.2                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  OCHF.sub. 2                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  OCHF.sub.2                                                                            2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            2-fluorocyclopropyl                                                                        Cl  OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  OCHF.sub.2                                                                            2,2-difluorocyclopropyl                                                                    Cl  OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  CH.sub.2 CN                                                                           cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           cyclopropyl CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  CH.sub.2 CN                                                                           cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           cyclopropyl OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           cyclopropyl Cl  OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  CH.sub.2 CN                                                                           cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           cyclobutyl  CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  CH.sub.2 CN                                                                           cyclobutyl  CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           cyclobutyl  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           cyclobutyl  Cl  OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           2-fluorocyclopropyl                                                                        Cl  OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            CH                                              H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                              H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           CH.sub.3                                                                            N                                               H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    OCH.sub.3                                                                          OCH.sub.3                                                                           N                                               H  CH.sub.2 CN                                                                           2,2-difluorocyclopropyl                                                                    Cl  OCH.sub.3                                                                           CH                                              __________________________________________________________________________

                                      TABLE VIII                                   __________________________________________________________________________                                       m.p.                                         R.sub.1                                                                          n R.sub.2                                                                              R'         X    Y    Z  (°C.)                                 __________________________________________________________________________     H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 Cl    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 Cl    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 Cl    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 Cl    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 Cl    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 Cl    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 Cl    cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 Cl    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 Cl    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 Cl    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 Cl    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 Cl    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 Cl    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 Cl    cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 Cl    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 Cl    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 Cl    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 Cl    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 Cl    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 Cl    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 Cl    cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 Cl    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 Cl    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 Cl    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 Cl    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 Cl    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 Cl    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 Cl    2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 CN    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CN    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CN    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CN    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CN    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CN    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CN    cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CN    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CN    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CN    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CN    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CN    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CN    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CN    cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 CN    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CN    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CN    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CN    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CN    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CN    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CN    cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CN    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CN    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CN    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CN    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CN    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CN    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CN    2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH CH.sub.3                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub. 3                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub. 3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 N(CH.sub.3).sub.2                                                                    CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH(CH.sub.3).sub.2                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH(CH.sub.3).sub.2                                                                        Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH(CH.sub.3).sub.2                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 CH.sub.3                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 CH(CH.sub.3).sub.2                                                      Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 Br                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 Br                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 Br                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 Br                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 Br                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 Br                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 Br                                                                      Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH(CH.sub.3)CH.sub.2 F                                                                    Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH(CH.sub.2 F).sub.2                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH(CH.sub.2 F).sub.2                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH(CH.sub.2 F).sub.2                                                                      Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 I CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 I CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 I OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 I CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 F                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 F                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 CH.sub.2 F                                                              Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 OCH.sub.2 F                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 OCH.sub.2 F                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 OCH.sub.2 F                                                                      Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 SOCH.sub.3                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 SOCH.sub.3                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 SOCH.sub.3                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SO.sub. 2 CH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 SO.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 SO.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 SO.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CN                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH.sub.2 CN                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 (CH.sub.3)CN                                                                     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 NO.sub.2                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 NO.sub.2                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CN                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CN                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 N(CH.sub.3).sub.2                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 N(CH.sub.3).sub.2                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH═ CH.sub.2                                                                 CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH═CH.sub.2                                                                  CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH═CH.sub.2                                                                  OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH═CH.sub.2                                                                  Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH═CH.sub.2                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH═CH.sub.2                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH═CH.sub.2                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH═CH.sub.2                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH═CH.sub.2                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH═CH.sub.2                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH═CH.sub.2                                                                           Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub. 3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub. 3                                                                          CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              __________________________________________________________________________

                                      TABLE IX                                     __________________________________________________________________________                                       m.p.                                         R.sub.1                                                                          n R.sub.2                                                                              R'         X    Y    Z  (°C.)                                 __________________________________________________________________________     H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CH.sub.3                                                                             2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CO CH.sub.3                                                                          cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 CO.sub.2 CH.sub.3                                                                    2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclobutyl Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCHF.sub.2                                                                           2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            CH.sub. 3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 SCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 F CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 F CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 F OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 F CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 F CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 F OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 F Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 F                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 H     CHF.sub.2  CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CHF.sub.2  CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CHF.sub.2  OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CHF.sub.2  CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CHF.sub.2  CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CHF.sub.2  OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CHF.sub.2  Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 Cl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 Cl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 Cl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 Cl                                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 OCH.sub.3                                                                        Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH(OCH.sub.3).sub.2                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH(OCH.sub.3).sub.2                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH(OCH.sub.3).sub.2                                                                       Cl   OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 0 H     CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 0 H     CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 0 H     CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 0 H     CH.sub.2 SCH.sub.3                                                                        Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.3   Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub. 2 CH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                              H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                               H 1 H     CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                              __________________________________________________________________________

                  TABLE X                                                          ______________________________________                                                                                       m.p.                             R.sub.1                                                                            n     R.sub.2  R'         X     Y     Z   (°C.)                     ______________________________________                                         H   0     H        cyclopropyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        cyclopropyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        cyclopropyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        cyclopropyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        cyclopropyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     H        cyclopropyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        cyclopropyl                                                                               Cl    OCH.sub.3                                                                            CH                                   H   0     H        cyclobutyl CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        cyclobutyl CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        cyclobutyl OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        cyclobutyl CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        cyclobutyl CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     H        cyclobutyl OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        cyclobutyl Cl    OCH.sub.3                                                                            CH                                   H   0     H        cyclopentyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        cyclopentyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        cyclopentyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        cyclopentyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        cyclopentyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     H        cyclopentyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        cyclopentyl                                                                               Cl    OCH.sub.3                                                                            CH                                   H   0     H        2-fluorocyclo-                                                                            CH.sub.3                                                                             CH.sub.3                                                                             CH                                                      propyl                                                      H   0     H        2-fluorocyclo-                                                                            CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     H        2-fluorocyclo-                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     H        2-fluorocyclo-                                                                            CH.sub.3                                                                             CH.sub.3                                                                             N                                                       propyl                                                      H   0     H        2-fluorocyclo-                                                                            CH.sub.3                                                                             OCH.sub.3                                                                            N                                                       propyl                                                      H   0     H        2-fluorocyclo-                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                       propyl                                                      H   0     H        2-fluorocyclo-                                                                            Cl    OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CH.sub.3 cyclopropyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 cyclopropyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclopropyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclopropyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 cyclopropyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 cyclopropyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 cyclopropyl                                                                               Cl    OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclobutyl CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 cyclobutyl CH.sub. 3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclobutyl OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclobutyl CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 cyclobutyl CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 cyclobutyl OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 cyclobutyl Cl    OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclopentyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 cyclopentyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclopentyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 cyclopentyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 cyclopentyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 cyclopentyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 cyclopentyl                                                                               Cl    OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 2-fluorocyclo-                                                                            CH.sub.3                                                                             CH.sub.3                                                                             CH                                                      propyl                                                      H   0     CH.sub.3 2-fluorocyclo-                                                                            CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CH.sub.3 2-fluorocyclo-                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CH.sub.3 2-fluorocyclo-                                                                            CH.sub.3                                                                             CH.sub.3                                                                             N                                                       propyl                                                      H   0     CH.sub.3 2-fluorocyclo-                                                                            CH.sub.3                                                                             OCH.sub.3                                                                            N                                                       propyl                                                      H   0     CH.sub.3 2-fluorocyclo-                                                                            OCH.sub.3                                                                            OCH.sub. 3                                                                           N                                                       propyl                                                      H   0     CH.sub.3 2-fluorocyclo-                                                                            Cl    OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclopropyl                                                                               Cl    OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclobutyl Cl    OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclopentyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CO.sub. 2 CH.sub.3                                                                      cyclopentyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclopentyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       cyclopentyl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclopentyl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclopentyl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CO.sub.2 CH.sub.3                                                                       cyclopentyl                                                                               Cl    OCH.sub.3                                                                            CH                                   H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            CH.sub.3                                                                             CH.sub.3                                                                             CH                                                      propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            CH.sub.3                                                                             OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            CH.sub.3                                                                             CH.sub.3                                                                             N                                                       propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            CH.sub.3                                                                             OCH.sub.3                                                                            N                                                       propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                            N                                                       propyl                                                      H   0     CO.sub.2 CH.sub.3                                                                       2-fluorocyclo-                                                                            Cl    OCH.sub.3                                                                            CH                                                      propyl                                                      H   0     CH.sub.3 CH.sub.3   CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 CH.sub.3   CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.3   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.3   CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 CH.sub.3   CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.3   OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.3   Cl    OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.3                                                                         Cl    OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl    OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     CH.sub.3 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl    OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 F CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        CH.sub.2 F CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 F OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 F CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        CH.sub.2 F CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 F OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 F Cl    OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        CH.sub.2 CH.sub.2 F                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 CH.sub.2 F                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 CH.sub.2 F                                                                       Cl    OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 F CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        CH.sub.2 F CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 F OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 F CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        CH.sub.2 F CH.sub. 3                                                                            OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 F OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 F Cl    OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                             CH.sub.3                                                                             CH                                   H   0     H        CH.sub.2 CF.sub.3                                                                         CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 CF.sub.3                                                                         OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   H   0     H        CH.sub.2 Cl                                                                               CH.sub.3                                                                             CH.sub.3                                                                             N                                    H   0     H        CH.sub.2 Cl                                                                               CH.sub.3                                                                             OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 Cl                                                                               OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    H   0     H        CH.sub.2 Cl                                                                               Cl    OCH.sub.3                                                                            CH                                   ______________________________________                                    

                                      TABLE XI                                     __________________________________________________________________________                                          m.p.                                      R.sub.1                                                                          n  R.sub.2 R'         X    Y    Z  (°C.)                              __________________________________________________________________________     H 0  H       cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  H       cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       cyclobutyl Cl   OCH.sub.3                                                                           CH                                           H 0  H       cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  CH.sub.3                                                                               cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  CH.sub.3                                                                               cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  CH.sub.3                                                                               cyclobutyI CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  CH.sub.3                                                                               cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               cyclobutyl Cl   OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  CH.sub.3                                                                               cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  CH.sub.3                                                                               cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               2-fluorocy-                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                                        clopropyl                                                         H 0  CH.sub.3                                                                               2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub. 3                                                                          CH                                           H 0  CH.sub.3                                                                               2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  CH.sub.3                                                                               2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  CH.sub.3                                                                               2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  CH.sub.3                                                                               2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclobutyl Cl   OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     cyclopentyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  OCH.sub.2 CF.sub.3                                                                     2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                           H 1  H       cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       cyclopropyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       cyclopropyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       cyclopropyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       cyclopropyl                                                                               Cl   OCH.sub.3                                                                           CH                                           H 1  H       cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       cyclobuty  OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 1  H       cyclobutyl CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       cyclobutyl CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       cyclobutyl OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       cyclobutyl Cl   OCH.sub.3                                                                           CH                                           H 1  H       cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 1  H       cyclopentyl                                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       cyclopentyl                                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       cyclopentyl                                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       cyclopentyI                                                                               Cl   OCH.sub.3                                                                           CH                                           H 1  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 1  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       2-fluorocyclopropyl                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       2-fluorocyclopropyl                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       2-fluorocyclopropyl                                                                       Cl   OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.3   Cl   OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub. 3                                                                          CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  SO.sub.2 N(CH.sub.3).sub.2                                                             CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.3   Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH  CH                                           H 0  H       CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.2 OCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 OCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 OCH.sub.3                                                                        Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 OCH.sub.2 CH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 OCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 CH.sub.2 OCH.sub.3                                                               CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH(OCH.sub.3).sub.2                                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH(OCH.sub.3).sub.2                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH(OCH.sub.3).sub.2                                                                       Cl   OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 0  H       CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 0  H       CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 0  H       CH.sub.2 SCH.sub.3                                                                        CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 SCH.sub.3                                                                        OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 0  H       CH.sub.2 SCH.sub.3                                                                        Cl   OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.3   CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       CH.sub.3   CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       CH.sub.3   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       CH.sub.3   Cl   OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       CH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       CH.sub.2 CH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       CH.sub.2 CH.sub.3                                                                         Cl   OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       CH.sub.2 CH.sub.2 CH.sub.3                                                                Cl   OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub. 3                                                                          CH                                           H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            CH.sub.3                                                                            N                                            H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                            OCH.sub.3                                                                           N                                            H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                            H 1  H       CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       Cl   OCH.sub.3                                                                           CH                                           __________________________________________________________________________

                  TABLE XII                                                        ______________________________________                                         J    R      R'       A    X.sub.1  Y.sub.1                                                                             m.p. (°C.)                      ______________________________________                                         J-1  CH.sub.3                                                                              CH.sub.3 A-2  CH.sub.3 O                                           J-1  CH.sub.3                                                                              CH.sub.3 A-2  OCH.sub.3                                                                               O                                           J-1  CH.sub.3                                                                              CH.sub.3 A-2  OCH.sub.2 CH.sub.3                                                                      O                                           J-1  CH.sub.3                                                                              CH.sub.3 A-2  OCF.sub.2 H                                                                             O                                           J-1  CH.sub.3                                                                              CH.sub.3 A-2  CH.sub.3 CH.sub.2                                    J-1  CH.sub.3                                                                              CH.sub.3 A-2  OCH.sub.3                                                                               CH.sub.2                                    J-2  --     cyclo-   A-2  CH.sub.3 O                                                       propyl                                                             J-2  --     cyclo-   A-2  OCH.sub.3                                                                               O                                                       propyl                                                             J-2  --     cyclo-   A-2  OCH.sub.2 CH.sub.3                                                                      O                                                       propyl                                                             J-2  --     cyclo-   A-2  OCF.sub.2 H                                                                             O                                                       propyl                                                             J-2  --     cyclo-   A-2  CH.sub.3 CH.sub.2                                                propyl                                                             J-2  --     cyclo-   A-2  OCH.sub.3                                                                               CH.sub.2                                                propyl                                                             J-3  --     cyclo-   A-2  CH.sub.3 O                                                       propyl                                                             J-3  --     cyclo-   A-2  OCH.sub.3                                                                               O                                                       propyl                                                             J-3  --     cyclo-   A-2  OCH.sub.2 CH.sub.3                                                                      O                                                       propyl                                                             J-3  --     cyclo-   A-2  OCF.sub.2 H                                                                             O                                                       propyl                                                             J-3  --     cyclo-   A-2  CH.sub.3 CH.sub.2                                                propyl                                                             J-3  --     cyclo-   A-2  OCH.sub.3                                                                               CH.sub.2                                                propyl                                                             ______________________________________                                         J    R       R'        A     X.sub.1  m.p. (°C.)                        ______________________________________                                         J-1  CH.sub.3                                                                               CH.sub.3  A-3   CH.sub.3                                          J-1  CH.sub.3                                                                               CH.sub.3  A-3   OCH.sub.3                                         J-1  CH.sub.3                                                                               CH.sub.3  A-3   OCH.sub.2 CH.sub.3                                J-1  CH.sub.3                                                                               CH.sub.3  A-3   OCF.sub.2 H                                       J-2  --      cyclo-    A-3   CH.sub.3                                                       propyl                                                            J-2  --      cyclo-    A-3   OCH.sub.3                                                      propyl                                                            J-2  --      cyclo-    A-3   OCH.sub.2 CH.sub.3                                             propyl                                                            J-2  --      cyclo-    A-3   OCF.sub.2 H                                                    propyl                                                            J-3  --      cyclo-    A-3   CH.sub.3                                                       propyl                                                            J-3  --      cyclo-    A-3   OCH.sub.3                                                      propyl                                                            J-3  --      cyclo-    A-3   OCH.sub.2 CH.sub.3                                             propyl                                                            J-3  --      cyclo-    A-3   OCF.sub.2 H                                                    propyl                                                            ______________________________________                                         J    R      R'       A    X.sub.1  Y.sub.3                                                                             m.p. (°C.)                      ______________________________________                                         J-1  CH.sub.3                                                                              CH.sub.3 A-4  CH.sub.3 H                                           J-1  CH.sub.3                                                                              CH.sub.3 A-4  OCH.sub. 3                                                                              H                                           J-1  CH.sub.3                                                                              CH.sub.3 A-4  OCH.sub.2 CH.sub.3                                                                      H                                           J-1  CH.sub.3                                                                              CH.sub.3 A-4  OCF.sub.2 H                                                                             H                                           J-1  CH.sub.3                                                                              CH.sub.3 A-4  CH.sub.3 CH.sub.3                                    J-1  CH.sub.3                                                                              CH.sub.3 A-4  OCH.sub.3                                                                               CH.sub.3                                    J-2  --     cyclo-   A-4  CH.sub.3 H                                                       propyl                                                             J-2  --     cyclo-   A-4  OCH.sub.3                                                                               H                                                       propyl                                                             J-2  --     cyclo-   A-4  OCH.sub.2 CH.sub.3                                                                      H                                                       propyl                                                             J-2  --     cyclo-   A-4  OCF.sub.2 H                                                                             H                                                       propyl                                                             J-2  --     cyclo-   A-4  CH.sub.3 CH.sub.3                                                propyl                                                             J-2  --     cyclo-   A-4  OCH.sub.3                                                                               CH.sub.3                                                propyl                                                             J-3  --     cyclo-   A-4  CH.sub.3 H                                                       propyl                                                             J-3  --     cyclo-   A-4  OCH.sub.3                                                                               H                                                       propyl                                                             J-3  --     cyclo-   A-4  OCH.sub.2 CH.sub.3                                                                      H                                                       propyl                                                             J-3  --     cyclo-   A-4  OCF.sub.2 H                                                                             H                                                       propyl                                                             J-3  --     cyclo-   A-4  CH.sub.3 CH.sub.3                                                propyl                                                             J-3  --     cyclo-   A-4  OCH.sub.3                                                                               CH.sub.3                                                propyl                                                             ______________________________________                                         J   R      R'       A    X.sub.2                                                                                Y.sub.2 m.p. (°C.)                     ______________________________________                                         J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.3                                                                              OCH.sub.3                                      J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.3                                                                              OCH.sub.2 CH.sub.3                             J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.3                                                                              SCH.sub.3                                      J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.3                                                                              CH.sub.3                                       J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.3                                                                              CH.sub.2 CH.sub.3                              J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                      J-1 CH.sub.3                                                                              CH.sub.3 A-5  CH.sub.2 CF.sub.3                                                                     CH.sub.3                                       J-2 --     cyclo-   A-5  CH.sub.3                                                                              OCH.sub.3                                                 propyl                                                              J-2 --     cyclo-   A-5  CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                        propyl                                                              J-2 --     cyclo-   A-5  CH.sub.3                                                                              SCH.sub.3                                                 propyl                                                              J-2 --     cyclo-   A-5  CH.sub.3                                                                              CH.sub.3                                                  propyl                                                              J-2 --     cyclo-   A-5  CH.sub.3                                                                              CH.sub.2 CH.sub.3                                         propyl                                                              J-2 --     cyclo-   A-5  CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                 propyl                                                              J-2 --     cyclo-   A-5  CH.sub.2 CF.sub.3                                                                     CH.sub.3                                                  propyl                                                              J-3 --     cyclo-   A-5  CH.sub.3                                                                              OCH.sub.3                                                 propyl                                                              J-3 --     cyclo-   A-5  CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                        propyl                                                              J-3 --     cyclo-   A-5  CH.sub.3                                                                              SCH.sub.3                                                 propyl                                                              J-3 --     cyclo-   A-5  CH.sub.3                                                                              CH.sub.3                                                  propyl                                                              J-3 --     cyclo-   A-5  CH.sub.3                                                                              CH.sub.2 CH.sub.3                                         propyl                                                              J-3 --     cyclo-   A-5  CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                 propyl                                                              J-3 --     cyclo-   A-5  CH.sub.2 CF.sub.3                                                                     CH.sub.3                                                  propyl                                                              ______________________________________                                         J     R       R'        A     X.sub.3 m.p. (°C.)                        ______________________________________                                         J-1   CH.sub.3                                                                               CH.sub.3  A-6   CH.sub.3                                         J-1   CH.sub.3                                                                               CH.sub.3  A-6   OCH.sub.3                                        J-2   --      cyclo-    A-6   CH.sub.3                                                       propyl                                                           J-2   --      cyclo-    A-6   OCH.sub.3                                                      propyl                                                           J-3   --      cyclo-    A-6   CH.sub.3                                                       propyl                                                           J-3   --      cyclo-    A-6   OCH.sub.3                                                      propyl                                                           ______________________________________                                         J    R      R'       A     X.sub.4                                                                               Y.sub.4                                                                              m.p. (°C.)                      ______________________________________                                         J-1  CH.sub.3                                                                              CH.sub.3 A-7   CH.sub.3                                                                              OCH.sub.3                                    J-1  CH.sub.3                                                                              CH.sub.3 A-7   OCH.sub.3                                                                             OCH.sub.3                                    J-2  --     cyclo-   A-7   CH.sub.3                                                                              OCH.sub.3                                                propyl                                                             J-2  --     cyclo-   A-7   OCH.sub.3                                                                             OCH.sub. 3                                               propyl                                                             J-3  --     cyclo-   A-7   CH.sub.3                                                                              OCH.sub.3                                                propyl                                                             J-3  --     cyclo-   A-7   OCH.sub.3                                                                             OCH.sub.3                                                propyl                                                             ______________________________________                                    

                  TABLE XIII                                                       ______________________________________                                         Compounds of Formula I where W = O, A is A-1, E is CH.sub.2,                   R is CH.sub.3 and n' is O                                                                                                     m.p.                            J   R.sub.1                                                                               R.sub.2                                                                              n   R'       X     Y     Z    (°C.)                    ______________________________________                                         J-8 H      H     1   CH.sub.3 CH.sub.3                                                                             CH.sub.3                                                                             CH                                   J-8 H      H     1   CH.sub.3 CH.sub.3                                                                             OCH.sub.3                                                                            CH                                   J-8 H      H     1   CH.sub.3 OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   J-8 CH.sub.3                                                                              H     1   CH.sub.3 OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   J-8 H      H     1   CH.sub.3 OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    J-8 H      H     1   CH.sub.3 OCH.sub.3                                                                            CH.sub.3                                                                             N                                    J-8 H      H     1   CH.sub.2 CH.sub.3                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH                                   J-8 H      H     1   CH.sub.2 CH.sub.3                                                                       OCH.sub.3                                                                            CH.sub.3                                                                             CH                                   J-8 H      H     1   CH.sub.2 CH.sub.3                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   J-8 H      H     1   CH.sub.2 CH.sub.3                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                            N                                    J-8 H      H     1   CH.sub.2 CH.sub.3                                                                       OCH.sub. 3                                                                           CH.sub.3                                                                             N                                    J-9 H      H     1   CH.sub.2 CH.sub.2 CH.sub.3                                                              OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   J-1 H      H     --  CH.sub.3 OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   J-6 H      H     --  CH.sub.3 OCH.sub.3                                                                            OCH.sub.3                                                                            CH                                   ______________________________________                                    

Formulations

Useful formulations of the compounds of Formula I can be prepared in conventional ways. They include dusts, granules, pellets, solutions, suspensions, emulsions, wettable powders, emulsifiable concentrates and the like. Many of these may be applied directly. Sprayable formulations can be extended in suitable media and used at spray volumes of from a few liters to several hundred liters per hectare. High strength compositions are primarily used as intermediates for further formulation. The formulations, broadly, contain about 0.1% to 99% by weight of active ingredient(s) and at least one of (a) about 0.1% to 20% surfactant(s) and (b) about 1% to 99.9% solid or liquid inert diluent(s). More specifically, they will contain these ingredients in the following approximate proportions:

    ______________________________________                                                     Active  Weight Percent*                                                        Ingredient                                                                             Diluent(s)                                                                               Surfactant(s)                                    ______________________________________                                         Wettable Powders                                                                             20-90      0-74     1-10                                         Oil Suspensions,                                                                              3-50     40-95     0-15                                         Emulsions, Solutions,                                                          (including Emulsifiable                                                        Concentrates)                                                                  Aqueous Suspension                                                                           10-50     40-84     1-20                                         Dusts          1-25     70-99     0-5                                          Granules and Pellets                                                                         0.1-95      5-99.9  0-15                                         High Strength 90-99      0-10     0-2                                          Compositions                                                                   ______________________________________                                          *Active ingredient plus at least one of a Surfactant or a Diluent equals       100 weight percent.                                                      

Lower or higher levels of active ingredient can, of course, be present depending on the intended use and the physical properties of the compound. Higher ratios of surfactant to active ingredient are sometimes desirable, and are achieved by incorporaton into the formulation or by tank mixing.

Typical solid diluents are described in Watkins, et al., "Handbook of Insecticide Dust Diluents and Carriers", 2nd Ed., Dorland Books, Caldwell, N.J., but other solids, either mined or manufactured, may be used. The more absorptive diluents are preferred for wettable powders and the denser ones for dusts. Typical liquid diluents and solvents are described in Marsden, "Solvents Guide," 2nd Ed., Interscience, New York, 1950. Solubility under 0.1% is preferred for suspension concentrates; solution concentrates are preferably stable against phase separation at 0° C. "McCutcheon's Detergents and Emulsifiers Annual", MC Publishing Corp., Ridgewood, N.J., as well as Sisely and Wood, "Encyclopedia of Surface Active Agents", Chemical Publishing Co., Inc., New York, 1964, list surfactants and recommended uses. All formulations can contain minor amounts of additives to reduce foaming, caking, corrosion, microbiological growth, etc.

The methods of making such compositions are well known. Solutions are prepared by simply mixing the ingredients. Fine solid compositions are made by blending and, usually, grinding as in a hammer or fluid energy mill. Suspensions are prepared by wet milling (see, for example, Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made by spraying the active material upon preformed granular carriers or by agglomeration techniques. See J. E. Browning, "Agglomeration", Chemical Engineering, Dec. 4, 1967, pp. 147ff. and "Perry's Chemical Engineer's Handbook", 5th Ed., McGraw-Hill, New York, 1973, p. 8-57ff.

For further information regarding the art of formulation, see for example:

H. M. Loux, U.S. Pat. No. 3,235,361, Feb. 15, 1966, Col. 6, line 16 through Col. 7, line 19 and Examples 10 through 41;

R. W. Luckenbaugh, U.S. Pat. No. 3,309,192, Mar. 14, 1967, Col. 5, line 43 through Col. 7, line 62 and Examples 8, 12, 15, 39, 41, 52, 53, 58, 132, 138-140, 162-164, 166, 167 and 169-182;

H. Gysin and E. Knusli, U.S. Pat. No. 2,891,855, June 23, 1959, Col. 3, line 66 through Col. 5, line 17 and Examples 1-4;

G. C. Klingman, "Weed Control as a Science", John Wiley and Sons, Inc., New York, 1961, pp. 81-96; and

J. D. Fryer and S. A. Evans, "Weed Control Handbook", 5th Ed., Blackwell Scientific Publications, Oxford, 1968, pp. 101-103.

In the following Examples, all parts are by weight unless otherwise indicated.

EXAMPLE 8

    ______________________________________                                          Wettable Powder                                                               ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      80%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       sodium alkylnaphthalenesulfonate                                                                             2%                                               sodium ligninsulfonate        2%                                               synthetic amorphous silica    3%                                               kaolinite                    13%                                               ______________________________________                                    

The ingredients are blended, hammer-milled until all the solids are essentially under 50 microns, reblended, and packaged.

EXAMPLE 9

    ______________________________________                                          Wettable Powder                                                               ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      50%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       sodium alkylnaphthalenesulfonate                                                                             2%                                               low viscosity methyl cellulose                                                                               2%                                               diatomaceous earth           46%                                               ______________________________________                                    

The ingredients are blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in diameter. The product is reblended before packaging.

EXAMPLE 10

    ______________________________________                                          Granule                                                                       ______________________________________                                         Wettable Powder of Example 9                                                                               5%                                                 attapulgite granules       95%                                                 (U.S.S. 20 to 40 mesh; 0.84-0.42 mm)                                           ______________________________________                                    

A slurry of wettable powder containing 25% solids is sprayed on the surface of attapulgite granules in a double-cone blender. The granules are dried and packaged.

EXAMPLE 11

    ______________________________________                                          Extruded Pellet                                                               ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      25%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       anhydrous sodium sulfate     10%                                               crude calcium ligninsulfonate                                                                                5%                                               sodium alkylnaphthalenesulfonate                                                                             1%                                               calcium/magnesium bentonite  59%                                               ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled.

EXAMPLE 12

    ______________________________________                                          Low Strength Granule                                                          ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                       0.1%                                             yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       attapulgite granules         99.9%                                             (U.S.S. 20 to 40 mesh)                                                         ______________________________________                                    

The active ingredient is dissolved in a solvent and the solution is sprayed upon dedusted granules in a double-cone blender. After spraying of the solution has been completed, the material is warmed to evaporate the solvent. The material is allowed to cool and then packaged.

EXAMPLE 13

    ______________________________________                                          Granule                                                                       ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      80%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       wetting agent                 1%                                               crude ligninsulfonate salt (containing                                                                      10%                                               5 to 20% of the natural sugars)                                                attapulgite clay              9%                                               ______________________________________                                    

The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the water content is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range. generally 14 to 100 mesh (1410 to 149 microns), and packaged for use.

EXAMPLE 14

    ______________________________________                                          Low Strength Granule                                                          ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                       1%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       N,N--dimethylformamide        9%                                               attapulgite granules         90%                                               (U.S.S. 20 to 40 sieve)                                                        ______________________________________                                    

The active ingredient is dissolved in the solvent and the solution is sprayed upon dedusted granules in a double cone blender. After spraying of the solution has been completed, the blender is allowed to turn for a short period and then the granules are packaged.

EXAMPLE 15

    ______________________________________                                          Aqueous Suspension                                                            ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      40%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       polyacrylic acid thickener   0.3%                                              dodecylphenol polyethylene glycol ether                                                                     0.5%                                              disodium phosphate           1%                                                monosodium phosphate         0.5%                                              polyvinyl alcohol            1.0%                                              water                        56.7%                                             ______________________________________                                    

The ingredients are blended and ground together in a sand mill to produce particles essentially all under 5 microns in size.

EXAMPLE 16

    ______________________________________                                          Solution                                                                      ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                       5%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide, ammonium                             salt                                                                           water                        95%                                               ______________________________________                                    

The salt is added directly to the water with stirring to produce the solution, which may then be packaged for use.

EXAMPLE 17

    ______________________________________                                          High Strength Concentrate                                                     ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                       99%                                              yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       silica aerogel               0.5%                                              synthetic amorphous silica   0.5%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce a material essentially all passing a U.S.S. No. 50 screen (0.3 mm opening). The concentrate may be formulated further if necessary.

EXAMPLE 18

    ______________________________________                                          Wettable Powder                                                               ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                       90%                                              yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       dioctyl sodium sulfosuccinate                                                                               0.1%                                              synthetic fine silica        9.9%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce particles essentially all below 100 microns. The material is sifted through a U.S.S. No. 50 screen and then packaged.

EXAMPLE 19

    ______________________________________                                          Wettable Powder                                                               ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      40%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       sodium ligninsulfonate       20%                                               montmorillonite clay         40%                                               ______________________________________                                    

The ingredients are thoroughly blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in size. The material is reblended and then packaged.

EXAMPLE 20

    ______________________________________                                          Oil Suspension                                                                ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      35%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       blend of polyalcohol carboxylic                                                                              6%                                               esters and oil soluble petroleum                                               sulfonates                                                                     xylene                       59%                                               ______________________________________                                    

The ingredients are combined and ground together in a sand mill to produce particles essentially all below 5 microns. The product can be used directly, extended with oils, or emulsified in water.

EXAMPLE 21

    ______________________________________                                          Dust                                                                          ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      10%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       attapulgite                  10%                                               Pyrophyllite                 80%                                               ______________________________________                                    

The active ingredient is blended with attapulgite and then passed through a hammer-mill to produce particles substantially all below 200 microns. The ground concentrate is then blended with powdered pyrophyllite until homogeneous.

EXAMPLE 22

    ______________________________________                                          Oil Suspension                                                                ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbon-                                                      25%                                               yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       polyoxyethylene sorbitol hexaoleate                                                                          5%                                               highly aliphatic hydrocarbon oil                                                                            70%                                               ______________________________________                                    

The ingredients are ground together in a sand mill until the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water.

EXAMPLE 23

    ______________________________________                                          Wettable Powder                                                               ______________________________________                                         4-Acetyl-N--[(4,6-dimethoxypyrimidin-2-yl)-[aminocarbon-                                                     20%                                              yl]-1-methyl-1-H--pyrazole-5-sulfonamide                                       sodium alkylnaphthalenesulfonate                                                                              4%                                              sodium ligninsulfonate         4%                                              low viscosity methyl celluose  3%                                              attapulgite                   69%                                              ______________________________________                                    

The ingredients are thoroughly blended. After grinding in a hammer-mill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) and packaged.

Utility

Test results indicate that the compounds of the present inventin are highly active preemergent or postemergent herbicides or plant growth regulants. Many of them have utility for broad-spectrum pre- and/or post-emergence weed control in areas where complete control of all vegetation is desired, such as around fuel shortage tanks, ammunition depots, industrial storage areas, parking lots, drive-in theaters, around billboards, highway and railroad structures. Some of the compounds have utility for selective weed control in crops such as wheat, barley, rice, soybeans and corn. Alternatively, the subject compounds are useful to modify plant growth.

The rates of application for the compounds of the invention are determined by a number of factors, including their use as plant growth modifiers or as herbicies, the crop species involved, the types of weeds to be controlled, weather and climate, formulations selected, mode of application, amount of foliage present, etc. In general terms, the subject compounds should be applied at levels of around 0.001 to 10 kg/ha, the lower rates being suggested for use on lighter soils and/or those having a low organic matter content, for plant growth modification or for situations where only short-term persistence is required.

The compounds of the invention may be used in combination with any other commercial herbicide, examples of which are those of the triazine, triazole, imidazolinone, uracil, urea, amide, diphenylether, carbamate and bipyridylium types as well as other sulfonylureas. They are particularly useful with the following herbicides.

    ______________________________________                                         Common Name                                                                              Chemical Name                                                        ______________________________________                                         alachlor  2-chloro-2',6'-diethyl-N--(methoxymethyl)-                                     acetanilide                                                          atrazine  2-chloro-4-(ethylamino)-6-(isopropylamino)-                                    s-triazine                                                           butylate  S--ethyl-diisobutylthiocarbamate                                     cyanazine 2-[[4-chloro-6-(ethylamino)-s-triazin-2-yl)-                                   amino]-2-methylpropionitrile                                         dicamba   3,6-dichloro-o-anisic acid                                           EPTC      S--ethyl dipropylthiocarbamate                                       linuron   3-(3,4-dichlorophenyl)-1-methoxy-1-                                            methylurea                                                           metolachlor                                                                              2-chloro-N--(2-ethyl-6-methylphenyl)-N--                                       (2-methoxy-1-methylethyl)acetamide                                   metribuzin                                                                               4-amino-6-tert-butyl-3-(methylthio)-as-                                        triazine-5(4H)--one                                                  tridiphane                                                                               2-(3,5-dichlorophenyl)-2-(2,2,2-tri-                                           chloroethyl)oxirane                                                  2,4-D     (2,4-dichlorophenoxy)acetic acid                                     thiobencarb                                                                              S--4-chlorobenzyldiethylthiocarbamate                                molinate  S--ethyl N,N--hexamethylenethiocarbamate                             butachlor N--(butoxymethyl)-2-chloro-2',6'-di-                                           ethylacetanilide                                                     naproanilide                                                                             N--phenyl-2-(1-naphthyloxy)propionamide                              pyrazolate                                                                               4-(2,4-dichlorobenzoyl)-1,3-dimethyl-                                          pyrazol-5-yl-4-toluenesulfonate                                      pretilachlor                                                                             2-chloro-2',6'-diethyl-N--(n-propoxy-                                          ethyl)acetanilide                                                    oxidiazon 3-[2,4-dichloro-5-(1-methylethoxy)-                                            phenyl]-5-(1,1-dimethylethyl)-1,3,4-                                           oxadiazol-2(3H)--one                                                 ______________________________________                                         Trade Name or                                                                  Code Number                                                                              Chemical Name                                                        ______________________________________                                         Harmony ®                                                                            3-[[(4-methoxy-6-methyl-1,3,5-triazin-                                         2-yl)aminocarbonyl]aminosulfonyl]-2-                                           thiophenecarboxylic acid, methyl ester                               Cinch ®                                                                              exo-1-methyl-4-(1-methylethyl)-2-[(2-                                          methylphenyl)methoxy]-7-oxabicyclo-                                            [2,2,1]heptane                                                       MY-93     S--(1-methyl-1-phenethyl)piperidine-1-                                         carbothioate                                                         CH-83     S--(2-methylpropyl)-hexanhydro-1H--aze-                                        pine-1-carbothioic acid, ester                                       X-52      2,4-dichlorophenyl-3-methoxy-4-nitro-                                          phenyl ether                                                         SC-2957   S---benzyl-N--ethyl-N--propylthiocarbamate                           HW-52     N--(2,3-dichlorophenyl)-4-(ethoxy-                                             methoxy)benzamide                                                    NTN-801   2-(benzothiazol-2-yl)-N--methyl-N--                                            phenylacetamide                                                      SL-49     2-[4-[(2.4-dichlorophenyl)carbonyl]-                                 20        1,3-dimethyl-1H--pyrazoI-5-yloxy]-1-                                           phenylethanone                                                       BAS-514   3,7-dichloro-8-quinoline carboxylic                                            acid                                                                 ______________________________________                                    

The herbidical properties of the subject compounds were discovered in a number of greenhouse tests. The test procedures and results follow.

    ______________________________________                                         Compounds                                                                      ______________________________________                                          ##STR47##                                                                     Compound   R'          X        Y      Z                                       ______________________________________                                         1          CH.sub.3    OCH.sub.3                                                                               OCH.sub.3                                                                             CH                                      2          CH.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3 CH.sub.3                                                                              CH                                      3          CH.sub.2 CH.sub.2 CH.sub.3                                                                 OCH.sub.3                                                                               CH.sub.3                                                                              CH                                      4          CH.sub.2 CH.sub.2 CH.sub.3                                                                 OCH.sub.3                                                                               OCH.sub.3                                                                             CH                                      5          CH.sub.2 CH.sub.2 CH.sub.3                                                                 OCH.sub.3                                                                               CH.sub.3                                                                              N                                       6          CH.sub.2 CH.sub.2 CH.sub.3                                                                 OCH.sub.3                                                                               OCH.sub.3                                                                             N                                       7          CH.sub.2 CH.sub.2 CH.sub.3                                                                 Cl       OCH.sub.3                                                                             CH                                      8          CH.sub.2 CH.sub.2 CH.sub.3                                                                 OCH.sub.3                                                                               OCH.sub.3                                                                             CH                                      9          CH.sub.2 CH.sub.3                                                                          CH.sub.3 CH.sub.3                                                                              CH                                      10         CH.sub.2 CH.sub.3                                                                          CH.sub.3 OCH.sub.3                                                                             CH                                      11         CH.sub. 2 CH.sub.3                                                                         CH.sub.3 OCH.sub.3                                                                             N                                       12         CH.sub.2 CH.sub.3                                                                          OCH.sub.3                                                                               OCH.sub.3                                                                             N                                       13         CH.sub.2 CH.sub.3                                                                          Cl       OCH.sub.3                                                                             CH                                      14         CH(CH.sub.3).sub.2                                                                         CH.sub.3 CH.sub.3                                                                              CH                                      15         CH(CH.sub.3).sub.2                                                                         CH.sub.3 OCH.sub.3                                                                             CH                                      16         CH(CH.sub.3).sub.2                                                                         OCH.sub.3                                                                               OCH.sub.3                                                                             CH                                      17         CH(CH.sub.3).sub.2                                                                         CH.sub.3 OCH.sub.3                                                                             N                                       18         CH(CH.sub.3).sub.2                                                                         OCH.sub.3                                                                               OCH.sub.3                                                                             N                                       19         CH(CH.sub.3).sub.2                                                                         Cl       OCH.sub.3                                                                             CH                                      ______________________________________                                          ##STR48##                                                                     Compound      X          Y          Z                                          ______________________________________                                         20            CH.sub.3   CH.sub.3   CH                                         21            CH.sub.3   OCH.sub.3  CH                                         22            OCH.sub.3  OCH.sub.3  CH                                         23            CH.sub.3   OCH.sub.3  N                                          24            OCH.sub.3  OCH.sub.3  N                                          25            Cl         OCH.sub.3  CH                                         ______________________________________                                    

Test A

Seeds of crabgrass (Digitaria spp.), barnyardgrass (Echinochloa crusgalli), giant foxtail (Setaria faberi), wild oats (Avena fatua), cheat grass (Bromus secalinus), velvetleaf (Abutilon theophrasti), morningglory (Ipomoea spp. ), cocklebur (Xanthium pennsylvanicum), sorghum, corn soybean, sugarbeet, cotton, rice, wheat, barley and purple nutsedge (Cyperus rotundus) tubers were planted and treated preemergence with the test chemicals dissolved in a non-phytotoxic solvent. At the same time, these crop and weed species were treated with a soil/foliage application. At the time of treatment, the plants ranged in height from 2 to 18 cm. Treated plants and controls were maintained in a greenhouse for sixteen days, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table A, are based on a numerical scale extending from 0=no injury, to 10=complete kill. The accompanying descriptive symbols have the following meanings:

C=chlorosis/necrosis

B=burn

D=defoliation

E=emergence inhibition

G=growth retardation

H=formative effect

U=unusual pigmentation

X=axillary stimulation

S=albinism

6Y=abscised buds or flowers

    TABLE A       Compound 1 Compound 2 Compound 3 Compound 4 Compound 5 Compound 6      Compound 7 Compound 8 Rate g/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE Corn 9H 3C,5H 0 0 3C,9H 1C,4H 3C,9H 3C,9H 2C,6H 0 6H 0 0      0 9C 4C,9G Wheat 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Barley 5G 0 0 0 2C 0 0      0 0 0 0 0 0 0 0 0 Rice 5C,9G 8G 4G 0 7G 3G 7G 2G 5G 3G 4C,9G 3G 2G 0 5G      0 Soybean 4C,9G 6H 0 0 2C,4H 1H 3C,8G,7X 3H 0 0 0 0 1C 0 3C,8H 3C,5H      Cotton 9G 9H 3C,8H 3C,8H 10C 4C,8H 4C,9G 4C,9G 8G 0 4C,9G 3G 7G 0 10C      10C Sugar Beet 9C 9C 3C,6G 2C,3G 4C,9H 3C,6G 4C,8G 4C,8G 1C 2G 3C,5G 2H      3C,6G 0 10C 10C Crabgrass 3C,8G 2C,6G 0 0 2G 0 4G 0 0 0 0 0 0 0 3C,7G 2G      Barnyardgrass 9C 5C,9H 2C,6G 0 4C,9H 2C,5G 5C,9H 3C,5H 2C,5H 2H 9H 0 0 0      9C 5C,9H Nutsedge 3C,9G 9G 7G 0 4C,9G 2C,5G 4C,9G 4C,8G 0 0 4G 0 0 0 9C      9C Giant Foxtail 5C,9G 3C,8G 2G 0 3C,7G 2G 4C,8G 4G 2G 0 2C,5G 0 0 0 10C      9C Cheatgrass 4C,9G 8G 6G 0 8G 5G 8G 2G 5G 0 5G 0 0 0 9C 7G Wild Oats      2C,5G 0 0 0 1C 0 0 0 0 0 0 0 0 0 0 0 Cocklebur 9C 3C,9H 4C,9G 3C,9H 9C      4C,9G 10C 6C,9G 5C,9G 4C,9H 4C,9G 4C,9H 3C,9G 2C,8H 10C 10C Morningglory      9C 3C,9H 3C,8G 2H 9C 3C,8G 10C 9C 4C,9G 3C,7G 5C,9G 3C,8H 3C,8G 3G 10C      10C Velvetleaf 9C 3C,8H 4C,9G 3G 9C 4C,9G 10C 4C,9G 3C,8H 2C,5G 3C,8H 6G      7G 0 9C 9C Sorghum             -- -- 3C,8H 3G PREEMERGENCE Corn 3C,9H      3C,7H 0 0 3C,8G 2C,7G 3C,8G 2C,6G 3C,6G 2C,4G 2C,5G 2C,5G 2C,3G 0 2C,9G      2C,9G Wheat 3G 0 0 0 0 0 0 0 0 0 0 0 0 0 2G 0 Barley 2C,5G 2C,4G 0 0 2G      0 0 0 0 0 5G 0 0 0 3G 0 Rice 9H 8H 2C 0 2C,2G 0 3G 0 4G 3G 2C,6G 2G      2C,3G 0 8H 2G Soybean 3C,6H 3C,4H 0 0 1H 0 3G 0 0 0 0 0 0 0 6H 6G Cotton      9G 6H 7G 5G 9G 8G 9G 8G 2C,2G 0 8G 2C,2G 5G 0 9G 9G Sugar beet 9G 4C,8G      0 0 8G 5G 9G 6G 4H 5G 9G 5G 8G 0 9G 8H Crabgrass 5G 2C,5G 0 0 0 0 0 0 0      0 0 0 0 0 2G 0 Barnyardgrass 9H 9H 2G 0 3C,7G 2G 3C,8G 2C,2G 3G 0 6G      2C,2G 3C,5G 0 9H 4G Nutsedge 10E 10E 0 0 7G 8G 9G 7G 0 0 0 0 0 0 10E 10E      Giant Foxtail 7G 3C,7H 0 0 2C,4G 0 3C,7G 0 4G 0 0 0 0 0 9H 5G Cheatgrass      9H 9H 0 0 4G 0 6G 0 0 0 5G 0 0 0 9G 8G Wild Oats 3G 2G 0 0 0 0 0 0 0 0 0      0 0 0 1C 0 Cocklebur 2C,7H 5H 8H 8H 9H 9H 9H 9H 7G 7H 9H 3H 9H -- 8H      3C,6H Morningglory 8H 8G 2G 0 9G 8G 8G 8G 6G 5G 7G 5H 8H 0 9H 9G      Velvetleaf 7H 0 5G 0 9C 9G 9C 9G 9C 8G 8G 3G 7G 0 8H 6H Sorghum         -- -- 9H 7G        CMPD 9 CMPD 10 CMPD 11 CMPD 12 CMPD 13 CMPD 14 CMPD 15 CMPD 16 CMPD 17 R      ATE RATE = KG/HA 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05        POSTEMERGENCE Cotton 10C 9C 10C 10C 7G 10C 6G 10C 10C 10C 3C,8G  9H      5C,9G  3C,6G Morningglory 3C,8G 9C 5C,9G 9C 4C,8H 10C 3C,8H 10C 4C,9G      10C 3C,6G  3C,8G  9C  3C,7H Cocklebur 10C 10C 10C 10C 5C,9G 10C 3C,7H 9C      9C 10C 3C,7G  4C,9G  10C  5C,9G Nutsedge 4C,9G 9C 5C,9G 9C 2G 3C,8G 0 0      4C,9G 10C 0  3C,8G  5C,9G  3C,5G Crabgrass 0 3G 3G 9C 0 4G 0 0 4G 0  0      2G  0 Barnyard Grass 3C,9H 9C 4C,9H 9C 6H 4C,9H 3H 4C,9H 7H 5C,9H 1C  0      3C,5H  0 Wild Oats 0 3C,6G 0 2C,6G 0 0 0 1C 0 0 0  0  0  0 Wheat 0 7G 0      7G 0 0 0 0 0 0 0  0  0  0 Corn 4G 2C,9H 9H 9C 9H 9G 3H 3C,9G 7H 3C,9G 0      7H  9G  8H Soybean 3H 6H 2C,3H 3C,7G 0 2H 0 7H 0 3G 2H  3C,5H  3H  1H      Rice 8G 9C 4G 2C,7G 2G 3C,9G 5G 6C,9G 2G 7G 3G  2G  1C  3G Sorghum 3C,9G      9C 4C,9H 9C 2C,9H 2C,9G 3C,8H 4C,9G 5G 3C,9H 3C,5G  3C,8H  3C,8G  3C,8G      Cheatgrass 2C,8G 9C 7G 9C 5G 5C,9G 0 4C,9G 5G 5C,9G 0  2G  2C,6G  3G      Sugar Beets 9C 10C 5C,9G 10C 5G 4C,8G 2H 6G 3C,7G 9C 3C,8G  5C,9G  5C,9G       4C,8G Velvet leaf 4C,9H 10C 9C 10C 2G 3C,8H 0 3C,7G 5G 3C,7G 3C,7G      4C,9G  9C  2C,5G 5G Giant Foxtail 2C,5G 5C,9G 3C,8G 9C 0 3C,7H 0 4G 5G      5C,9H 1C  2G  4G  2C Barley 6G 3C,8G 0 3C,7G 0 0 0 0 0 3G 0  0  0  0      PREEMERGENCE Cotton 8H 9G 8G 9G 0 8H 0 5G 3G 8G 0  2G  7G  0 Morningglory       7H 9G 9G 9G 0 9G 0 7H 7G 9G 0  3C,4H  9G  2C,5G Cocklebur 9H 9H 9H  1C      2C,7H 1H 3C,3H 3H  0  3C,5G  3C,7H  2C Nutsedge 9G 9G 8G 10E 0 10E 0 0      7G 9G 0  10E  9G  0 Crabgrass 0 0 0 4G 0 0 0 0 0 3G 0    8G  0 Barnyard      Grass 7G 9H 6H 9H 0 7H 0 3H 2G 9H 0  0  2G  0 Wild Oats 0 2G 2C 2C,4G 0      0 0 0 0 0 0  0  0  0 Wheat 0 4G 0 3G 0 0 0 2G 0 0 0  0  0  0 Corn 0      2C,9G 3C,9H 9H 2C,9H 2C,9G 4H 2C,9H 2C,5G 9G 0  2C  3C,4G  3C,6G Soybean      3G 5G 3G 2C,7H 0 3C,4G 0 1C,1H 0 2G 0  1H  3G  0 Rice 8H 9H 7G 3C,8H 7H      9H 8G 9H 0 8G 0  0  2G  0 Sorghum 9H 10H 9H 10H 9G 9H 2C,7H 5C,9G 3C,8H      3C,9H 0  2C  5G  3C,5G Cheatgrass 5G 9G 8G 9G 0 9H 0 3G 5G 9G 0  0  4G      0 Sugar Beets 9G 9G 4C,9G 3C,9G 7H 3C,8G 4H 5G 8G 9G 3G  3G  8G  7G      Velvetleaf 5H 9H 8H 9H 0 2H 0 2C,2G 3H 7H 0  2C,2H  6H  2C Giant Foxtail      0 2G 2C,4G 8G 0 3G 0 0 0 7G 0  0  5G  0 Barley 7G 2C,8G 0 7G 0 6G 2G 5G      0 2C,3G 0  0  0  0        CMPD 18 CMPD 19 CMPD 20 CMPD 21 CMPD 22  CMPD 23 CMPD 24 CMPD 25 RATE      RATE = KG/HA 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0      .01 0.05 0.01 0.05        POSTEMERGENCE Cotton 3C,6H  2G  4C,9G 5C,9G 5C,9G 9C 3C,9G 4C,9G 9C      10C 4C,9G 4C,9G 9C 9C Morningglory 3C,7G  2C,4H  3H 10C 10C 10C 4C,9G      10C 10C 10C 10C 10C 10C 10C Cocklebur 4C,8H  3C,7G  5C,9G 9C 9C 10C 10C      10C 10C 10C 10C 10C 9C 10C Nutsedge 0  0  3C,8G 4C,9G 4C,8G 9C 9C 10C 0      0 0 2C,5G 9C 9C Crabgrass 0  0  0 0 0 4G 0 3G 0 0 0 0 0 0 Barnyard Grass      0  0  3C,7H 4C,9H 3C,9H 9C 3C,5G 3C,8H 0 3C,7H 0 5H 0 2H Wild Oats 0  0      3G 3C,8G 5G 7G 0 3G 0 2G 0 2G 0 0 Wheat 0  0  3G 2C,7G 3G 7G 3G 4G 0 3G      0 3G 0 2G Corn 3C,8H  0  2G 7H 8H 3C,9H 2G 3C,9H 2C,3G 9H 0 4G 0 0      Soybean 1H  0  5H 3C,8G 5C,9G 4C,9G 3C,9G 4C,9G 9C 5C,9G 4C,9G 4C,9G 0      8G Rice 7G  0  8G 5C, 9G 7G 3C, 9G 4G 2C, 8G 2G 4C, 8G 1C 4C, 8G 4H 3G      Sorghum 3C,8G  3C,5G  4C,9H 9C 9H 10C 7H 3C,9H 3G 3C,8H 2C,3G 2C,6H 0      3C,8G Cheatgrass 2G  0  3C,7G 3C,9G 5C,9G 5C,9G 3C,5G 9C 0 2G 0 2C,4G 0      3G Sugar Beets 4C,9H  2C,3G  4C,8G 4C,8G 10C 10C 9C 10C 9C 9C 10C 9C 4G      10C Velvetleaf 3C,6G  1C  10C 9C 10C 10C 4C,9G 10C 10C 10C 2C,4H 5G 9C      10C Giant Foxtail 1C  0  2G 3C,3G 3G 3C,8G 0 2C,4H 0 3G 0 3C,5G 0 0      Barley 0  0  3G 9G 5G 8G 2G 4G 0 3G 0 0 0 0 PREEMERGENCE Cotton 0  0  2G      8G 7G 8H 0 5G 8H 9G 5G 3C,8G 0 2G Morningglory 2C  2C  0 6G 5G 9G 2G 7G      9G 9G 9G 4C,9G 5G 9H Cocklebur 2C  1C  3G 9H 4H 3C,6H 2G 7G 3C,7H 9H      3C,8H 9H  1C Nutsedge 0 0  0 0  6G 0 10E 0 0 0 0 5G 9G Crabgrass 4G  4G      0 0 0 4G 0 2G 0 0 0 0 0 0 Barnyard Grass 0  0  7G 8H 7H 9H 0 7H 1C 2H 0      0 0 4H Wild Oats 0  0  2G 7H 2G 3C,8G 0 0 0 0 0 0 0 0 Wheat 0  0  0 7G      2G 7G 0 0 0 0 0 0 0 0 Corn 2C,5G  0  0 7H 2C,8H 9G 0 3C,7G 3C,4G 3C,7G      1C 2C,5G 0 2G Soybean 0  0  2G 3C,3H 3C,5G 3C,9H 1C,1H 3C,5H 3C,7H 9G      3C,7H 3C,9H 0 1C Rice 3G 0  8G 9H 8G 3C,9H 7G 9G 0 8G 3G 7G 0 7G Sorghum      2C,3G  2C,4G  9H 10H 3C,9H 3C,9H 8G 3C,9H 2C,3G 8G 2C, 3G 3C,6G 3G 2C,7G      Cheatgrass 0  0  5G 8G 5G 9G 0 8G 0 2G 0 0 0 3G Sugar Beets 7H  4G  5H      7G 3C,8G 5C,9G 2G 3C,7G 9C 9G 4C,9G 9C 5G 8G Velvetleaf 2G  0  5G 8H 6H      9G 0 4H 7H 4C,9G 0 2G 3G 6H Giant Foxtail 2G  0  0 0 2G 4H 0 4G 0 0 0 0      0 0 Barley 0  0  0 7G 2G 2C,8G 0 1C 0 2C,3G 0 1C 0 0

Test B Postemergence

Three round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with nutsedge (Cyperus rotundus) rubers, crabgrass (Digitaria sanguinalis), sicklepod (Cassia obtusifolia), jimsonweed (Datura stramonium), velvetleaf (Abutilon theophrasti), lambsquarters (Chenopodium album), rice (Oryza sativa) and teaweed (Sida spinosa). The second pot was planted with green foxtail (Setaria viridis), cocklebur (Xantium pensylvanicum), morningglory (Ipomoea hederacea), cotton (Gossypium hirsutum), johnsongrass (Sorghum halepense), barnyardgrass (Echinochloa crusgalli), corn (Zea mays), soybean (Glycine max) and giant foxtail (Setaria faberi). The third pot was planted with wheat (Triticum aestivum), barley (Hordeum vulgare), wild buckwheat (Polgonum convolvulus L.), cheatgrass (Bromus secalinus L.) sugarbeet (Beta vulgaris), wild oats (Avena fatua), viola (Viola arvensis), blackgrass, (Alopecurus myosuroides), and rape (Brassica napus). The plants were grown for approximately fourteen days, then sprayed postemergence with the chemicals dissolved in a non-phytotoxic solvent.

Preemergence

Three round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with nutsedge tubers, crabgrass, sickelpod, jimsonweed, velvetleaf, lambsquarters, rice and teaweed. The second pot was planted with green foxtail, cocklebur, morningglory, cotton, johnsongrass, barnyardgrass, corn, soybean and giant foxtail. The third pot was planted with wheat, barley, wild buckwheat, cheatgrass, sugarbeet, wild oat, viola, blackgrass and rape. The three pans were sprayed preemergence with the chemicals dissolved in a non-phytotoxic solvent.

Treated plants and controls were maintained in the greenhouse for 25 days, then all rated plants were compared to controls and visually rated for plant response.

Response ratings are based on a scale of 0 to 100 where 0=no effect and 100=complete control. A dash (--) response means no test.

Response ratings are contained in Table B.

                  TABLE B                                                          ______________________________________                                                  Compound 3                                                                      POSTEMER-                                                                     GENCE       PREEMERGENCE                                              Rate g/ha  62     16    4   1    250  62   16  4                               ______________________________________                                         Corn       20     0     0   0    40   0    0   0                               Wheat      0      0     0   0    0    0    0   0                               Barley     0      0     0   0    0    0    0   0                               Rice       0      0     0   0    60   40   20  0                               Soybean    0      0     0   0    20   0    0   0                               Cotton     70     50    30  0    50   20   0   0                               Sugar beet 100    70    50  30   100  90   80  70                              Rape       90     70    50  30   90   80   70  50                              Crabgrass  60     30    0   0    50   30   0   0                               Johnsongrass                                                                              70     30    0   0    90   70   50  30                              Blackgrass 30     0     0   0    70   30   0   0                               Barnyardgrass                                                                             70     30    0   0    80   60   40  0                               Nutsedge   80     60    30  0    0    0    0   0                               Giant Foxtail                                                                             30     0     0   0    80   60   40  0                               Green Foxtail                                                                             70     30    0   0    90   70   50  30                              Cheatgrass 30     0     0   0    90   60   30  0                               Wild Oats  0      0     0   0    0    0    0   0                               Wild Buckwheat                                                                            70     50    30  0    90   70   50  30                              Viola      90     70    50  30   100  90   70  50                              Lambsquarter                                                                              100    70    50  30   100  90   70  50                              Cocklebur  100    90    70  50   80   50   30  0                               Morningglory                                                                              100    70    50  30   90   60   30  0                               Teaweed    90     70    50  30   80   60   40  20                              Sicklepod  60     30    0   0    100  70   50  30                              Jimsonweed 70     50    30  0    90   70   50  30                              Velvetleaf 90     70    50  30   90   70   50  30                              ______________________________________                                                  Compound 4                                                                      POSTEMER-                                                                     GENCE       PREEMERGENCE                                              Rate g/ha  62     16    4   1    250  62   16  4                               ______________________________________                                         Corn       30     0     0   0    60   20   0   0                               Wheat      0      0     0   0    30   0    0   0                               Barley     0      0     0   0    30   0    0   0                               Rice       0      0     0   0    70   30   0   0                               Soybean    20     0     0   0    0    0    0   0                               Cotton     90     40    0   0    20   0    0   0                               Sugar beet 100    90    70  50   100  90   70  50                              Rape       100    70    40  0    90   80   70  50                              Crabgrass  70     50    30  0    50   30   0   0                               Johnsongrass                                                                              50     30    0   0    70   50   30  0                               Blackgrass 0      0     0   0    30   0    0   0                               Barnyardgrass                                                                             90     60    30  0    70   30   0   0                               Nutsedge   90     70    50  30   100  70   50  30                              Giant Foxtail                                                                             80     60    30  0    70   50   30  0                               Green Foxtail                                                                             70     50    30  0    90   70   50  30                              Cheatgrass 30     0     0   0    70   30   0   0                               Wild Oats  100    70    50  30   0    0    0   0                               Wild Buckwheat                                                                            90     70    50  30   80   60   40  0                               Viola      100    90    70  50   100  90   70  50                              Lambsquarter                                                                              90     70    50  30   100  90   80  70                              Cocklebur  100    90    70  50   90   70   50  30                              Morningglory                                                                              100    90    70  50   90   80   60  40                              Teaweed    90     70    50  30   90   70   50  30                              Sicklepod  80     70    50  30   100  100  70  50                              Jimsonweed 100    70    50  30   90   70   50  30                              Velvetleaf 100    70    50  30   90   80   70  50                              ______________________________________                                                  Compound 4                                                                      POSTEMER-                                                                     GENCE       PREEMERGENCE                                              Rate g/ha  62     16    4   1    250  62   16  4                               ______________________________________                                         Corn       30     0     0   0    60   20   0   0                               Wheat      0      0     0   0    30   0    0   0                               Barley     0      0     0   0    30   0    0   0                               Rice       0      0     0   0    70   30   0   0                               Soybean    20     0     0   0    0    0    0   0                               Cotton     90     40    0   0    20   0    0   0                               Sugar beet 100    90    70  50   100  90   70  50                              Rape       100    70    40  0    90   80   70  50                              Crabgrass  70     50    30  0    50   30   0   0                               Johnsongrass                                                                              50     30    0   0    70   50   30  0                               Blackgrass 0      0     0   0    30   0    0   0                               Barnyardgrass                                                                             90     60    30  0    70   30   0   0                               Nutsedge   90     70    50  30   100  70   50  30                              Giant Foxtail                                                                             80     60    30  0    70   50   30  0                               Green Foxtail                                                                             70     50    30  0    90   70   50  30                              Cheatgrass 30     0     0   0    70   30   0   0                               Wild Oats  100    70    50  30   0    0    0   0                               Wild Buckwheat                                                                            90     70    50  30   80   60   40  0                               Viola      100    90    70  50   100  90   70  50                              Lasmbsquarter                                                                             90     70    50  30   100  90   80  70                              Cocklebur  100    90    70  50   90   70   50  30                              Morningglory                                                                              100    90    70  50   90   80   60  40                              Teaweed    90     70    50  30   90   70   50  30                              Sicklepod  80     70    50  30   100  100  70  50                              Jimsonweed 100    70    50  30   90   70   50  30                              Velvetleaf 100    70    50  30   90   80   70  50                              ______________________________________                                                      CMPD 8                                                            RATE RATE = G/HA                                                                              0004     0016    0062   0250                                    ______________________________________                                         PREEMERGENCE                                                                   GIANT FOXTAIL  40       90      100    100                                     VELVETLEAF     50       90      100    100                                     SUGAR BEETS    90       100     100    100                                     CRABGRASS      0        0       20     90                                      TEAWEED        30       80      90     100                                     JIMSONWEED     40       80      100    100                                     RICE           0        0       20     100                                     COCKLEBUR      40       50      90     100                                     COTTON         30       50      70     100                                     SOYBEAN        0        20      50     100                                     BARNYARD GRASS 50       90      100    100                                     WILD OATS      0        0       0      0                                       MORNINGGLORY   40       60      100    100                                     WHEAT          0        0       0      0                                       CASSIA         0        40      70     100                                     JOHNSONGRASS   0        40      60     90                                      NUTSEDGE       90       100     100    100                                     CORN           20       50      70     100                                     WILD BUCKWHEAT 80       90      100    100                                     BLACK GRASS             40      90     90                                      RAPESEED       40       90      100    100                                     BARLEY         0        0       0      0                                       GREEN FOXTAIL  70       100     100    100                                     CHEAT GRASS    70       90      90     100                                     LAMBSQUARTER   90       100     100    100                                     ______________________________________                                                      CMPD 8                                                            RATE RATE = G/HA                                                                              0001     0004    0016   0062                                    ______________________________________                                         POSTEMERGENCE                                                                  GIANT FOXTAIL  20       60      90     100                                     VELVETLEAF     100      100     100    100                                     SUGAR BEETS    70       80      100    100                                     CRABGRASS      0        20      50     100                                     TEAWEED        0        30      70     100                                     JIMSONWEED     0        50      100    100                                     RICE           0        0       0      0                                       COCKLEBUR      40       70      100    100                                     COTTON         40       40      80     90                                      SOYBEAN        20       40      60     70                                      BARNYARD GRASS 40       40      80     100                                     WILD OATS      0        0       0      20                                      MORNINGGLORY   0        30      80     100                                     WHEAT          0        0       0      0                                       CASSIA         30       30      50     100                                     JOHNSONGRASS   0        0       0      0                                       NUTSEDGE       80       100     100    100                                     CORN           0        20      80     90                                      WILD BUCKWHEAT 30       50      100    100                                     BLACK GRASS    0        0       30     30                                      RAPESEED       100      100     100    100                                     BARLEY         0        0       0      0                                       GREEN FOXTAIL  0        30      100    100                                     CHEAT GRASS    0        30      50     80                                      BUCKWHEAT                                                                      VIOLA                                                                          LAMBSQUARTER   100                     100                                     ______________________________________                                                      CMPD 22                                                           RATE RATE = G/HA                                                                              0001     0004    0016   0062                                    ______________________________________                                         POSTEMERGENCE                                                                  GIANT FOXTAIL  0        0       30     50                                      VELVETLEAF     50       70      100    100                                     SUGAR BEETS    70       80      90     90                                      CRABGRASS      0        0       30     70                                      TEAWEED        30       50      70     90                                      JIMSONWEED     30       50      70     100                                     RICE           0        20      30     50                                      COCKLEBUR      50       80      100    100                                     COTTON         50       60      70     80                                      SOYBEAN        70       90      90     100                                     BARNYARD GRASS 0        0       0      40                                      WILD OATS      0        0       0      0                                       MORNINGGLORY   60       80      100    100                                     WHEAT          0        0       0      0                                       CASSIA         30       50      80     100                                     JOHNSONGRASS   0        0       30     70                                      NUTSEDGE       30       40      60     100                                     CORN           0        0       20     60                                      WILD BUCKWHEAT 30       50      70     80                                      BLACK GRASS    0        0       30     50                                      RAPESEED       100      100     100    100                                     BARLEY         0        0       0      20                                      GREEN FOXTAIL  0        0       30     50                                      CHEAT GRASS    0        0       30     60                                      VIOLA          70       90      100    100                                     LAMBSQUARTER   30       40      50     70                                      ______________________________________                                                      CMPD 22                                                           RATE RATE = G/HA                                                                              0004     0016    0062   0250                                    ______________________________________                                         PREEMERGENCE                                                                   GIANT FOXTAIL  0        30      50     70                                      VELVETLEAF     30       50      70     90                                      SUGAR BEETS    70       80      90     100                                     CRABGRASS      0        30      60     90                                      TEAWEED        50       70      80     90                                      JIMSONWEED     50       70      80     90                                      RICE           30       50      80     100                                     COCKLEBUR      60       70      80     90                                      COTTON         0        30      50     70                                      SOYBEAN        0        20      40     60                                      BARNYARD GRASS 30       50      70     90                                      WILD OATS      0        0       20     30                                      MORNINGGLORY   70       80      90     100                                     WHEAT          0        0       0      0                                       CASSIA         30       50      70     90                                      JOHNSONGRASS   30       50      70     90                                      NUTSEDGE       50       70      100    100                                     CORN           0        0       20     60                                      WILD BUCKWHEAT 70       80      90     100                                     BLACK GRASS    50       60      70     80                                      RAPESEED       80       90      100    100                                     BARLEY         0        0       0      0                                       GREEN FOXTAIL  0        30      60     90                                      CHEAT GRASS    0        30      50     80                                      LAMBSQUARTER   70       80      90     100                                     ______________________________________                                    

Test C

Sixteen cm diameter Wagner pots, equipped with a stoppered drain opening near the bottom of the side wall, were partially filled with Woodstown sandy loam. About 1500 mls of water were added to each pot to bring the water level to a point 3 cm above the soil surface. Japonica and Indica rice seedlings were transplanted as described in Test E. Also, a number of barnyardgrass (Echinochola crusgalli) seeds were added to each pot. At the same time, seedlings or tubers of the following species were transplanted into the muddy soil: water plantain (Alisma trivale), Scirpus (Scirpus mucranatus), and Cyperus (Cyperus difformis). The weed species selected for this test are of economic importance in major rice-growing areas. The chemical treatments were applied directly to the paddy water after being formulated in a nonphytotoxic solvent within hours after transplanting of two additional species: water chestnuts (Eleocharis spp.) and arrowhead (Sagittaria latifolia). Shortly after treatment, the drain hole was opened to drop the water level by 2 cm. Water was then added to restore the water level to its original height. The following day the draining and refilling process was repeated. The pots were then maintained in the greenhouse. Rates of application and plant response ratings made 21 days after treatment are summarized in Table C.

In the subsequent tables, LS is used as an abbreviation for leaf stage.

                  TABLE C                                                          ______________________________________                                                       CMPD 8                                                           RATE RATE = G/HA                                                                               0004      0008     0016                                        ______________________________________                                         SOIL                                                                           BARNYARD GRASS  50        67       70                                          WATER CHESTNUT  62        77       90                                          ARROWHEAD       0         57       80                                          SCIRPUS (SEDGE) 37        72       85                                          CYPRESS (SEDGE) 75        75       95                                          WATER PLANTAIN  75        55       90                                          RICE JAP EFF    0         0        10                                          RICE INDICA EFF 0         17       0                                           ______________________________________                                    

Test D

The soybeans were planted in large 25 cm-diameter pots of soil, 6 to 10 plants per pot. The other plant species were planted in 15 cm-diamter pots of soil. Corn, because of its importance as a rotational crop, was by itself in one container, 3 to 5 plants per pot. The weed species used in this test were all of major economic importance in soybean-growing regions. They were planted 3 to 4 species per pot, each confined to a separate quadrant of the soil surface. The following species were included in the screen:

    ______________________________________                                         barnyardgrass     Echinochloa crus-galli                                       giant foxtail     Setaria faberi                                               green foxtail     Setaris virdis                                               johnsongrass      Sorghum halepense                                            fall panicum      Panicum dichotomiflorum                                      purple nutsedge   Cyperus rotundus                                             signalgrass       Brachiaria platyphylla                                       crabrass          Digitaria sanguinalis                                        velvetleaf        Abutilon theophrasti                                         jimsonweed        Datura stramonium                                            hemp sesbania     Sesbania exaltata                                            sicklepod         Cassia obtusifolia                                           cocklebur         Xanthium pensylvanicum                                       ivyleaf morninglory                                                                              Ipomoea hederacea                                            purslane          portulaca oleracea                                           pigweed           Amaranthus retroflexus                                       lambsquarter      Chenopodium album                                            teaweed           Sida spinosa                                                 bindweed          Convolvulus arvensis                                         ______________________________________                                    

For the post-emergence phase of the test, crop and weed species were planted two to three weeks before application so that they were present as young plants at the time of treatment. Plantings for the pre-emergence phase were made on the day before, or on the day of treatment. Approximate planting depths were: corn and soybean--3 to 4 cm; morningglory, cocklebur and nutsedge--2.5 to 3 cm; velvetleaf, sicklepod and sesbania--2 cm; all other species--0.5 cm.

The test chemicals were dissolved/suspended in a non-phytotoxic solvent in concentrations required to obtain the desirec rate of application. The solutions or suspensions were then applied as soil/foliage sprays to the young plants (post-emergence phase) and to the soil surfaces of the freshly planted containers (pre-emergence phase). Application was made utilizing an automatic spray machine at a spray volume of 500 liters per hectare. Immediately after treatment, the containers were transferred to a greenhouse and subsequently watered on a demand basis, taking care not to wet the foilage of the plants in the post-emergence phase of the test.

Visual plant response ratings were made approximately two and four weeks after treatment for the post- and pre-emergence phases, respectively. The ratings were made on a percentage scale of 0 to 100, where 0=no injury, and 100=death of plants, and are summarized in Table D.

                  TABLE D                                                          ______________________________________                                          COMPOUND 9                                                                    ______________________________________                                         RATE RATE GM/H                                                                               0002   0004     0008 0016   0031                                 ______________________________________                                         POSTEMERGENCE                                                                  SOYBEAN       0      0        0    20     60                                   CORN          0      0        0    50     70                                   VELVETLEAF    50     65       90   100    100                                  NIGHTSHADE    0      20       30   75     85                                   JIMSONWEED    0      0        20   30     40                                   SICKLEPOD     0      0        0    20     50                                   SESBANIA      0      0        0    30     50                                   COCKLEBUR     40     85       100  100    100                                  IVYLEAF M/G   30     65       75   80     95                                   PIGWEED       40     60       75   85     90                                   LAMBSQUARTER  30     60       85   85     85                                   PRICKLY SIDA  0      30       50   75     85                                   SMARTWEED     40     50       80   80     90                                   BARNYARDGRASS 0      30       50   70     80                                   GIANT FOXTAIL 0      0        0    40     65                                   GREEN FOXTAIL 0      0        0    40     60                                   JOHNSONGRASS  0      30       65   80     95                                   FALL PANICUM  0      20       40   50     75                                   CRABGRASS     0      0        0    20     30                                   SIGNALGRASS   0      20       30   50     65                                   NUTSEDGE      65     80       90   100    100                                  ______________________________________                                         RATE RATE GM/H  0031   0062      0125 0250                                     ______________________________________                                         PREEMERGENCE                                                                   SOYBEAN         0      0         25   60                                       CORN            0      20        65   90                                       VELVETLEAF      0      20        80   95                                       NIGHTSHADE      50     70        85   95                                       JIMSONWEED      0      30        70   95                                       SICKLEPOD       0      0         30   60                                       SESBANIA        0      0         40   50                                       COCKLEBUR       80     75        80   95                                       IVYLEAF M/G     0      0         40   50                                       PIGWEED         70     85        100  100                                      LAMBSQUARTER    20     75        95   100                                      PRICKLY SIDA    40     70        80   90                                       SMARTWEED       70     90        90   100                                      BARNYARDGRASS   0      0         40   85                                       GIANT FOXTAIL   0      0         30   70                                       GREEN FOXTAIL   0      20        40   70                                       JOHNSONGRASS    85     90        95   95                                       FALL PANICUM    90     100       100  95                                       CRABGRASS       0      0         20   40                                       SIGNALGRASS     0      30        70   85                                       NUTSEDGE        80     90        100  100                                      ______________________________________                                     

What is claimed:
 1. A compound of Formula I ##STR49## wherein J is ##STR50## R is H, C₁ -C₃ alkyl, phenyl, SO₂ NR_(a) R_(b), C₁ -C₂ haloalkyl, C₂ -C₄ alkoxyalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₄ alkylthioalkyl, C₂ -C₄ alkylsulfinylalkyl, C₂ -C₄ alkylsulfonylalkyl, CO₂ C₁ -C₂ alkyl, C₁ -C₄ alkylcarbonyl, C₁ -C₂ alkylsulfonyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl or C₁ -C₂ alkyl substituted with CO₂ C₁ -C₂ alkyl;R₁ is H or CH₃ ; R₂ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(c) R_(d), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, CO₂ R_(e), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₂ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio, CN, OH or SH; R_(a) and R_(b) are independently C₁ -C₂ alkyl; R_(c) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy; R_(d) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or R_(c) and R_(d) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --; R_(e) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl; R' is C₁ -C₅ alkyl, C₁ -C₅ haloalkyl, C₁ -C₅ alkyl substituted with one or two R₃ groups, C₂ -C₅ alkenyl, C₂ -C₅ haloalkenyl, C₃ -C₅ alkenyl substituted with one or two R₃ groups, C₃ -C₅ alkynyl, C₃ -C₅ haloalkynyl, C₃ -C₅ alkynyl substituted with one or two R₃ groups, C₃ -C₅ cycloalkyl, C₃ -C₅ halocycloalkyl, C₃ -C₅ cycloalkyl substituted with one or two R₄ groups, C₄ -C₇ cycloalkylalkyl, C₄ -C₇ halocycloalkylalkyl, C₄ -C₇ cycloalkylalkyl substituted with one or two R₄ groups, phenyl or benzyl; R₃ is C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₁ -C₃ haloalkoxy, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, NO₂, OH, OR₅ or di-(C₁ -C₃ alkyl)amino; R₄ is C₁ -C₃ alkyl, C₁ -C₃ alkoxy, C₁ -C₃ haloalkoxy, CN, NO₂, OH, OR₅ or di-(C₁ -C₃ alkyl)amino; R₅ is SO₂ CH₃, Si(CH₃)₃, C₂ -C₃ alkylcarbonyl or CO₂ C₁ -C₂ alkyl; E is a single bond or CH₂ ; W is O or S; n is O or 1; n' is 0 or 1; A is ##STR51## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl; Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, ##STR52## or N(OCH₃)CH₃ ; m is 2 or 3; L₁ and L₂ are independently O or S; R₆ is H or C₁ -C₃ alkyl; R₇ and R₈ are independently C₁ -C₃ alkyl; and Z is CH;and their agriculturally suitable salts; provided that (a) when X is Cl, F, Br or I, then Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H; (b) when W is S, then R₁ is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C═CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or 1,3-dioxolan-2-yl; (c) when the total number of carbons of X and Y is greater than four, then the number of carbons of R must be less than or equal to two; (d) when J is J-1 or J-2, then R' is other than C₃ -C₅ cycloalkyl or phenyl; (e) when J is J-5, J-6 or J-7 wherein E is a single bond, then R' is other than C₁ -C₅ alkyl, C₂ -C₅ alkenyl, phenyl, benzyl, cyclopentyl or C₄ -C₇ cycloalkylalkyl; (f) when either or both of X and Y are OCF₂ H then J is J-1, J-2, J-8, J-9, J-10 or J-11; and (g) when the total number of carbon atoms of X and Y is greater than four, then the total number of carbon atoms of R₂ and R' must be less than or equal to 7, (h) when J is J-5, J-6 or J-7 and E is CH₂, then R' is other than C₁ -C₅ alkyl.
 2. Compounds of claim 1 where E is a single bond; and W is O.
 3. Compounds of claim 1 where E is CH₂ ; and W is O.
 4. Compounds of claim 2 whereR₂ is H, C₁ -C₃ alkyl, halogen, C₁ -C₃ alkyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br, OCH₃, SO₂ NHCH₃, SO₂ N(CH₃)₂, S(O)_(n) CH₃, CO₂ CH₃, CO₂ CH₂ CH₃, OCF₂ H, CH₂ OCH₃ or CH₂ CN; R is H, C₁ -C₃ alkyl, phenyl, CH₂ CF₃ or CH₂ CH═CH₂ ; X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, Cl, F, Br, I, OCF₂ H, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ .tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR53## OCF₂ H, OCF₂ Br, SCF₂ H, cyclopropyl, C.tbd.CH or C.tbd.CCH₃.
 5. Compounds of claim 4 whereR' is C₁ -C₄ alkyl, C₁ -C₃ alkyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br, C₂ -C₄ alkoxyalkyl, C₂ -C₄ alkylthioalkyl, C₂ -C₄ cyanoalkyl, C₂ -C₄ alkenyl, C₂ -C₃ alkenyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br, C₃ -C₄ alkynyl, C₃ -C₅ cycloalkyl, C₃ -C₅ cycloalkyl substituted with 1 to 3 halogen atoms selected from 1 to 3 Cl, 1 to 3 F or 1 Br or cyclopropylmethyl.
 6. Compounds of claim 5 wheren is O; X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCF₂ H; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃, CH(OCH₃)₂ or cyclopropyl.
 7. Compounds of claim 6 whereR₁ is H; R₂ is H, Cl, Br, OCH₃ or CH₃ ; and R' is C₁ -C₃ alkyl, C₁ -C₃ alkyl substituted with 1 to 3 F, C₂ -C₃ alkoxyalkyl, C₂ -C₃ alkylthioalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₃ alkenyl, propargyl, C₃ -C₅ cycloalkyl or cyclopropylmethyl.
 8. Compounds of claim 7 where J is J-1.
 9. Compounds of claim 8 where R' is C₁ -C₃ alkyl.
 10. Compounds of claim 8 where R' is C₁ -C₃ alkyl substituted with 1 to 3 F, C₂ -C₃ alkoxyalkyl, C₂ -C₃ alkylthioalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₃ alkenyl, propargyl, C₃ -C₅ cyclo alkyl or cyclopropylmethyl.
 11. Compounds of claim 3 whereR is H, C₁ -C₃ alkyl, phenyl CH₂ CF₃ or CH₂ CH═CH₂ ; R₂ is H, Cl, Br, OCH₃ or CH₃ ; R' is C₁ -C₃ alkyl, C₁ -C₃ alkyl substituted with 1 to 3 F, C₂ -C₃ alkoxyalkyl, C₂ -C₃ alkylthioalkyl, C₂ -C₃ cyanoalkyl, C₂ -C₃ alkenyl, propargyl, C₃ -C₅ cycloalkyl or cyclopropylmethyl; n is O; X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCF₂ H; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃, CH(OCH₃)₂ or cyclopropyl.
 12. Compounds of claim 1 whereJ is J-1, J-2, J-3 or J-4; and R' is C₁ -C₅ haloalkyl, C₁ -C₅ alkyl substituted with one or two R₃ groups, C₂ -C₅ alkenyl, C₂ -C₅ haloalkenyl, C₃ -C₅ alkenyl substituted with one or two R₃ groups, C₃ -C₅ alkynyl, C₃ -C₅ haloalkynyl, C₃ -C₅ alkynyl substituted with one or two R₃ groups, C₃ -C₅ cycloalkyl, C₃ -C₅ halocycloalkyl, C₃ -C₅ cycloalkyl substituted with one or two R₄ groups, C₄ -C₇ cycloalkylalkyl substituted with one or two R₄ groups, phenyl or benzyl.
 13. Compounds of claim 1 which are 4-(1-oxopropyl)-N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-1H-pyrazole-5-sulfonamide.
 14. Compounds of claim 1 which are 2-(cyclopropylcarbonyl)-N-[4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-thiophenesulfonamide.
 15. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 1 and at least one of the following: surfactant, solid or liquid diluent.
 16. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 2 and at least one of the following: surfactant, solid or liquid diluent.
 17. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 3 and at least one of the following: surfactant, solid or liquid diluent.
 18. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 4 and at least one of the following: surfactant, solid or liquid diluent.
 19. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 5 and at least one of the following: surfactant, solid or liquid diluent.
 20. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 6 and at least one of the following: surfactant, solid or liquid diluent.
 21. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 7 and at least one of the following: surfactant, solid or liquid diluent.
 22. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 8 and at least one of the following: surfactant, solid or liquid diluent.
 23. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 9 and at least one of the following: surfactant, solid or liquid diluent.
 24. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 10 and at least one of the following: surfactant, solid or liquid diluent.
 25. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 11 and at least one of the following: surfactant, solid or liquid diluent.
 26. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 12 and at least one of the following: surfactant, solid or liquid diluent.
 27. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 13 and at least one of the following: surfactant, solid or liquid diluent.
 28. An agriculturally suitable composition for controlling the growth of undesired vegetation comprising an effective amount of the compound of claim 14 and at least one of the following: surfactant, solid or liquid diluent.
 29. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 1. 30. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 2. 31. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 3. 32. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 4. 33. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 5. 34. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 6. 35. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 7. 36. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 8. 37. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 9. 38. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 10. 39. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 11. 40. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 12. 41. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 13. 42. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 14. 